Literature summary for 3.5.3.15 extracted from

Trabocchi, A.; Pala, N.; Krimmelbein, I.; Menchi, G.; Guarna, A.; Sechi, M.; Dreker, T.; Scozzafava, A.; Supuran, C.; Carta, F.
Peptidomimetics as protein arginine deiminase 4 (PAD4) inhibitors (2015), J. Enzyme Inhib. Med. Chem., 30, 466-471 .

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Inhibitors

Inhibitors	Comment	Organism	Structure
(3R)-3-[2-[4-(2-carbamimidamidoethyl)-1H-1,2,3-triazol-1-yl]acetamido]-3-(4-fluorophenyl)propanoic acid	1,2,3-triazole peptidomimetic-based compound, 39% inhibition at 1 microM, 99% inhibition at 10 microM	Homo sapiens
(3S)-3-[2-[4-(2-carbamimidamidoethyl)-1H-1,2,3-triazol-1-yl]acetamido]-3-phenylpropanoic acid	1,2,3-triazole peptidomimetic-based compound, 26% inhibition at 1 microM, 69% inhibition at 10 microM	Homo sapiens

Organism

Organism	UniProt	Comment	Textmining
Homo sapiens	Q9UM07	-	-

Source Tissue

Source Tissue	Comment	Organism	Textmining
commercial preparation	-	Homo sapiens	-

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Release 2023.1 (January 2023)