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Literature summary for 3.5.1.88 extracted from

  • Antczak, C.; Shum, D.; Escobar, S.; Bassit, B.; Kim, E.; Seshan, V.E.; Wu, N.; Yang, G.; Ouerfelli, O.; Li, Y.M.; Scheinberg, D.A.; Djaballah, H.
    High-throughput identification of inhibitors of human mitochondrial peptide deformylase (2007), J. Biomol. Screen., 12, 521-535.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
2',2'-bisepigallocatechin monogallate
-
Homo sapiens
3-methoxycatechol
-
Homo sapiens
7,8-dihydroxyflavone
-
Homo sapiens
actinonin
-
Homo sapiens
chloranil
-
Homo sapiens
epigallocatechin 3,5-digallate
-
Homo sapiens
epitheaflavin monogallate
-
Homo sapiens
hematein
-
Homo sapiens
hematoxylin
-
Homo sapiens
irigenol
-
Homo sapiens
additional information development of a high-throughput assay to screen for inhibitors Homo sapiens
purpurogallin
-
Homo sapiens
pyrogallin
-
Homo sapiens
quinalizarin
-
Homo sapiens
theaflavin
-
Homo sapiens
theaflavin monogallate
-
Homo sapiens
thiram
-
Homo sapiens

Localization

Localization Comment Organism GeneOntology No. Textmining
mitochondrion
-
Homo sapiens 5739
-

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Homo sapiens

Synonyms

Synonyms Comment Organism
HsPDF
-
Homo sapiens

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.0027
-
fluorescence polarization assay Homo sapiens hematoxylin
0.0041
-
fluorescence polarization assay Homo sapiens 2',2'-bisepigallocatechin monogallate
0.0055
-
fluorescence polarization assay Homo sapiens actinonin
0.0057
-
fluorescence polarization assay Homo sapiens pyrogallin
0.0061
-
fluorescence polarization assay Homo sapiens theaflavin
0.0071
-
fluorescence polarization assay Homo sapiens theaflavin monogallate
0.0088
-
fluorescence polarization assay Homo sapiens purpurogallin
0.0089
-
fluorescence polarization assay Homo sapiens quinalizarin
0.012
-
fluorescence polarization assay Homo sapiens hematein
0.017
-
fluorescence polarization assay Homo sapiens 7,8-dihydroxyflavone
0.017
-
fluorescence polarization assay Homo sapiens irigenol
0.029
-
fluorescence polarization assay Homo sapiens epitheaflavin monogallate
0.031
-
fluorescence polarization assay Homo sapiens 3-methoxycatechol
0.038
-
fluorescence polarization assay Homo sapiens epigallocatechin 3,5-digallate
0.043
-
fluorescamine assay Homo sapiens thiram
0.048
-
fluorescence polarization assay Homo sapiens chloranil