Inhibitors | Comment | Organism | Structure |
---|---|---|---|
actinonin | IC50: 0.000043 mM | Homo sapiens | |
siRNA HsPDF 581-601 | transfection of HeLa cells | Homo sapiens | |
siRNA HsPDF 659-679 | transfection of HeLa cells | Homo sapiens | |
SKI-AC-1 | IC50: 0.000072 mM, actionin analog | Homo sapiens | |
SKI-AC-10 | IC50: 0.000078 mM, actionin analog | Homo sapiens | |
SKI-AC-11101 | IC50: 0.000076 mM, actionin analog | Homo sapiens | |
SKI-AC-111101 | IC50: 0.0000600 mM, actionin analog | Homo sapiens | |
SKI-AC-111110 | IC50: 0.000427 mM, actionin analog | Homo sapiens | |
SKI-AC-111111 | IC50: 0.000069 mM, actionin analog | Homo sapiens | |
SKI-AC-111112 | IC50: 0.000234 mM, actionin analog | Homo sapiens | |
SKI-AC-111113 | IC50: 0.000177 mM, actionin analog | Homo sapiens | |
SKI-AC-111114 | IC50: 0.000300 mM, actionin analog | Homo sapiens | |
SKI-AC-11112 | IC50: 0.000365 mM, actionin analog | Homo sapiens | |
SKI-AC-11113 | IC50: 0.000500 mM, actionin analog | Homo sapiens | |
SKI-AC-11114 | IC50: 0.000276 mM, actionin analog | Homo sapiens | |
SKI-AC-11115 | IC50: 0.000473 mM, actionin analog | Homo sapiens | |
SKI-AC-11116 | IC50: 0.000335 mM, actionin analog | Homo sapiens | |
SKI-AC-11117 | IC50: 0.000086 mM, actionin analog | Homo sapiens | |
SKI-AC-11118 | IC50: 0.000115 mM, actionin analog | Homo sapiens | |
SKI-AC-11119 | IC50: 0.000134 mM, actionin analog | Homo sapiens | |
SKI-AC-11128 | IC50: 0.000522 mM, actionin analog | Homo sapiens | |
SKI-AC-11138 | IC50: 0.000500 mM, actionin analog | Homo sapiens | |
SKI-AC-11148 | IC50: 0.0000600 mM, actionin analog | Homo sapiens | |
SKI-AC-11158 | IC50: 0.000500 mM, actionin analog | Homo sapiens | |
SKI-AC-11168 | IC50: 0.000192 mM, actionin analog | Homo sapiens | |
SKI-AC-11178 | IC50: 0.000200 mM, actionin analog | Homo sapiens | |
SKI-AC-11188 | IC50: 0.000120 mM, actionin analog | Homo sapiens | |
SKI-AC-11198 | IC50: 0.000090 mM, actionin analog | Homo sapiens | |
SKI-AC-3 | IC50: 0.000500 mM, actionin analog | Homo sapiens | |
SKI-AC-5 | IC50: 0.000400 mM, actionin analog | Homo sapiens | |
SKI-AC-51121 | IC50: 0.000400 mM, actionin analog | Homo sapiens | |
SKI-AC-6 | IC50: 0.000097 mM, actionin analog | Homo sapiens | |
SKI-AC-8 | IC50: 0.000093 mM, actionin analog | Homo sapiens | |
SKI-AC-9 | IC50: 0.000151 mM, actionin analog | Homo sapiens | |
SKI-AC-I-18 | IC50: 0.000404 mM, actionin analog | Homo sapiens | |
SKI-AC-I-19 | IC50: 0.000239 mM, actionin analog | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.45 | - |
formyl-Met-Thr-Met-His | - |
Homo sapiens | |
1.7 | - |
formyl-Met-Ala-His-Ala | - |
Homo sapiens | |
11 | - |
formyl-Met-Ala-Ser | - |
Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
mitochondrion | - |
Homo sapiens | 5739 | - |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
formyl-L-methionyl peptide + H2O | Homo sapiens | - |
formate + methionyl peptide | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | Q9HBH1 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
A-2780 cell | - |
Homo sapiens | - |
CWR22Rv1 cell | - |
Homo sapiens | - |
DAUDI cell | - |
Homo sapiens | - |
DU-145 cell | - |
Homo sapiens | - |
HEK-293 cell | - |
Homo sapiens | - |
HeLa cell | - |
Homo sapiens | - |
HL60 cell | - |
Homo sapiens | - |
HT-1080 cell | - |
Homo sapiens | - |
MDA-MB-468 cell | - |
Homo sapiens | - |
NB-4 cell | - |
Homo sapiens | - |
PBMC | - |
Homo sapiens | - |
PC3 cell | - |
Homo sapiens | - |
RAJI cell | - |
Homo sapiens | - |
RL cell | - |
Homo sapiens | - |
SK-BR-3 cell | - |
Homo sapiens | - |
SK-LC-16 cell | - |
Homo sapiens | - |
SK-LC-8 cell | - |
Homo sapiens | - |
Tsu-Pr1 cell | - |
Homo sapiens | - |
WI-38 cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
formyl-L-methionyl peptide + H2O | - |
Homo sapiens | formate + methionyl peptide | - |
? | |
formyl-Met-Ala-His-Ala + H2O | fMAHA | Homo sapiens | formate + methionyl-Ala-His-Ala | - |
? | |
formyl-Met-Ala-Ser + H2O | fMAS | Homo sapiens | formate + Met-Ala-Ser | - |
? | |
formyl-Met-Thr-Met-His + H2O | fMTMH | Homo sapiens | formate + methionyl-Thr-Met-His | - |
? |
Synonyms | Comment | Organism |
---|---|---|
HsPDF | - |
Homo sapiens |
- |
Homo sapiens | |
peptide deformylase | - |
Homo sapiens |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
25 | - |
activity assay | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.4 | - |
activity assay | Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.000043 | - |
IC50: 0.000043 mM | Homo sapiens | GLLI | |
0.00006 | - |
IC50: 0.0000600 mM, actionin analog | Homo sapiens | SKI-AC-111101 | |
0.00006 | - |
IC50: 0.0000600 mM, actionin analog | Homo sapiens | SKI-AC-11148 | |
0.000069 | - |
IC50: 0.000069 mM, actionin analog | Homo sapiens | SKI-AC-111111 | |
0.000072 | - |
IC50: 0.000072 mM, actionin analog | Homo sapiens | SKI-AC-1 | |
0.000076 | - |
IC50: 0.000076 mM, actionin analog | Homo sapiens | SKI-AC-11101 | |
0.000078 | - |
IC50: 0.000078 mM, actionin analog | Homo sapiens | SKI-AC-10 | |
0.000086 | - |
IC50: 0.000086 mM, actionin analog | Homo sapiens | SKI-AC-11117 | |
0.00009 | - |
IC50: 0.000090 mM, actionin analog | Homo sapiens | SKI-AC-11198 | |
0.000093 | - |
IC50: 0.000093 mM, actionin analog | Homo sapiens | SKI-AC-8 | |
0.000097 | - |
IC50: 0.000097 mM, actionin analog | Homo sapiens | SKI-AC-6 | |
0.000115 | - |
IC50: 0.000115 mM, actionin analog | Homo sapiens | SKI-AC-11118 | |
0.00012 | - |
IC50: 0.000120 mM, actionin analog | Homo sapiens | SKI-AC-11188 | |
0.000134 | - |
IC50: 0.000134 mM, actionin analog | Homo sapiens | SKI-AC-11119 | |
0.000151 | - |
IC50: 0.000151 mM, actionin analog | Homo sapiens | SKI-AC-9 | |
0.000177 | - |
IC50: 0.000177 mM, actionin analog | Homo sapiens | SKI-AC-111113 | |
0.000192 | - |
IC50: 0.000192 mM, actionin analog | Homo sapiens | SKI-AC-11168 | |
0.0002 | - |
IC50: 0.000200 mM, actionin analog | Homo sapiens | SKI-AC-11178 | |
0.000234 | - |
IC50: 0.000234 mM, actionin analog | Homo sapiens | SKI-AC-111112 | |
0.000239 | - |
IC50: 0.000239 mM, actionin analog | Homo sapiens | SKI-AC-I-19 | |
0.000276 | - |
IC50: 0.000276 mM, actionin analog | Homo sapiens | SKI-AC-11114 | |
0.0003 | - |
IC50: 0.000300 mM, actionin analog | Homo sapiens | SKI-AC-111114 | |
0.000335 | - |
IC50: 0.000335 mM, actionin analog | Homo sapiens | SKI-AC-11116 | |
0.000365 | - |
IC50: 0.000365 mM, actionin analog | Homo sapiens | SKI-AC-11112 | |
0.0004 | - |
IC50: 0.000400 mM, actionin analog | Homo sapiens | SKI-AC-5 | |
0.0004 | - |
IC50: 0.000400 mM, actionin analog | Homo sapiens | SKI-AC-51121 | |
0.000404 | - |
IC50: 0.000404 mM, actionin analog | Homo sapiens | SKI-AC-I-18 | |
0.000427 | - |
IC50: 0.000427 mM, actionin analog | Homo sapiens | SKI-AC-111110 | |
0.000473 | - |
IC50: 0.000473 mM, actionin analog | Homo sapiens | SKI-AC-11115 | |
0.0005 | - |
IC50: 0.000500 mM, actionin analog | Homo sapiens | SKI-AC-3 | |
0.0005 | - |
IC50: 0.000500 mM, actionin analog | Homo sapiens | SKI-AC-11113 | |
0.0005 | - |
IC50: 0.000500 mM, actionin analog | Homo sapiens | SKI-AC-11138 | |
0.0005 | - |
IC50: 0.000500 mM, actionin analog | Homo sapiens | SKI-AC-11158 | |
0.000522 | - |
IC50: 0.000522 mM, actionin analog | Homo sapiens | SKI-AC-11128 |