Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1,4-diaminobutane | Ki: 1.45 mM; putrescine | Rattus sp. | |
1,5-Diaminopentane | cadaverine; Ki: 1.5 mM | Rattus sp. | |
1,6-diaminohexane | Ki: 1.5 mM | Rattus sp. | |
acetylprocainamide | Ki: 1.9 mM | Rattus sp. | |
N1-acetylspermidine | Ki: 0.16 mM, competitive inhibition | Rattus sp. | |
spermidine | Ki: 0.31 mM | Rattus sp. | |
spermine | Ki: 1.15 mM | Rattus sp. |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.004 | - |
N8-Acetylspermidine | - |
Rattus sp. |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
cytosol | - |
Rattus sp. | 5829 | - |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus sp. | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
liver | - |
Rattus sp. | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
N8-acetylspermidine + H2O | involvement in controlling the levels of polyamines and acetylated polyamines in tissues | Rattus sp. | acetate + spermidine | - |
? |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.31 | - |
spermidine | - |
Rattus sp. | |
1.15 | - |
spermine | - |
Rattus sp. | |
1.45 | - |
1,4-diaminobutane | - |
Rattus sp. | |
1.5 | - |
1,6-diaminohexane | - |
Rattus sp. | |
1.5 | - |
1,5-Diaminopentane | - |
Rattus sp. | |
1.9 | - |
acetylprocainamide | - |
Rattus sp. |