Cloned (Comment) | Organism |
---|---|
expression in Sf9 cells | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
N-Boc-Cys(farnesyl)-methylenamin-VIM-OH | i.e. isoprenyl protease inhibitor RPI, 0.000058 mM, 50% inhibition | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.002 | - |
K-Ras(farnesyl)VIM | - |
Homo sapiens | |
0.003 | - |
2-aminobenzoyl-KSKTKC(farnesyl) | - |
Homo sapiens | |
0.003 | - |
2-aminobenzoyl-KSKTKC(farnesyl)lysine-epsilon-dinitrophenyl-IM | - |
Homo sapiens | |
0.004 | - |
KSKTKC(farnesyl)VIM | - |
Homo sapiens | |
0.004 | - |
7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl)VIM | - |
Homo sapiens | |
0.004 | - |
7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl)VI-lysine-epsilon-dinitrophenyl | - |
Homo sapiens | |
0.004 | - |
7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl)-dinitrophenyldiaminopropionic acid-IM | - |
Homo sapiens | |
0.004 | - |
2-aminobenzoyl-KSKTKC(farnesyl)VIM | - |
Homo sapiens | |
0.004 | - |
2-aminobenzoyl-KSKTKC(farnesyl)VI | - |
Homo sapiens | |
0.004 | - |
2-aminobenzoyl-KSKTKC(farnesyl)VI-dinitrophenyldiaminopropionic acid | - |
Homo sapiens | |
0.005 | - |
7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl)-VI-dinitrophenyldiaminopropionic acid | - |
Homo sapiens | |
0.005 | - |
2-aminobenzoyl-KSKTKC(farnesyl)VI-lysine-epsilon-dinitrophenyl | - |
Homo sapiens | |
0.006 | - |
7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl)lysine-epsilon-dinitrophenyl | - |
Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
membrane | - |
Homo sapiens | 16020 | - |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
35000 | - |
- |
Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
K-Ras(farnesyl)VIM + H2O | Homo sapiens | - |
K-Ras(farnesyl) + VIM | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
2-aminobenzoyl-KSKTKC(farnesyl)dinitrophenyldiaminopropionic acid-IM + H2O | 34% of activity with KSKTKC(farnesyl)VIM | Homo sapiens | 2-aminobenzoyl-KSKTKC(farnesyl) + dinitrophenyldiaminopropionic acid-IM | - |
? | |
2-aminobenzoyl-KSKTKC(farnesyl)lysine-epsilon-dinitrophenyl-IM + H2O | 50% of activity with KSKTKC(farnesyl)VIM | Homo sapiens | 2-aminobenzoyl-KSKTKC(farnesyl) + lysine-epsilon-dinitrophenyl-IM | - |
? | |
2-aminobenzoyl-KSKTKC(farnesyl)VI + H2O | - |
Homo sapiens | ? | - |
? | |
2-aminobenzoyl-KSKTKC(farnesyl)VI-dinitrophenyldiaminopropionic acid + H2O | 4.8% of activity with KSKTKC(farnesyl)VIM | Homo sapiens | 2-aminobenzoyl-KSKTKC(farnesyl) + VI-dinitrophenyldiaminopropionic acid | - |
? | |
2-aminobenzoyl-KSKTKC(farnesyl)VI-lysine-epsilon-dinitrophenyl + H2O | 25% of activity with KSKTKC(farnesyl)VIM | Homo sapiens | 2-aminobenzoyl-KSKTKC(farnesyl) + VI-lysine-epsilon-dinitrophenyl | - |
? | |
2-aminobenzoyl-KSKTKC(farnesyl)VIM + H2O | - |
Homo sapiens | 2-aminobenzoyl-KSKTKC(farnesyl) + VIM | - |
? | |
7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl)-dinitrophenyldiaminopropionic acid-IM + H2O | 2.5% of activity with KSKTKC(farnesyl)VIM | Homo sapiens | 7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl) + dinitrophenyldiaminopropionic acid-IM | - |
? | |
7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl)-VI-dinitrophenyldiaminopropionic acid + H2O | 1% of activity with KSKTKC(farnesyl)VIM | Homo sapiens | 7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl) + VI-dinitrophenyldiaminopropionic acid | - |
? | |
7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl)lysine-epsilon-dinitrophenyl + H2O | - |
Homo sapiens | 7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl) + lysine-epsilon-dinitrophenyl-IM | - |
? | |
7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl)VI-lysine-epsilon-dinitrophenyl + H2O | 2% of activity with KSKTKC(farnesyl)VIM | Homo sapiens | 7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl) + VI-lysine-epsilon-dinitrophenyl | - |
? | |
7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl)VIM + H2O | 35% of activity with KSKTKC(farnesyl)VIM | Homo sapiens | 7-methoxycoumarin-4-acetyl-KSKTKC(farnesyl) + VIM | - |
? | |
K-Ras(farnesyl)VIM + H2O | - |
Homo sapiens | K-Ras(farnesyl) + VIM | - |
? | |
KSKTKC(farnesyl)VIM + H2O | no activity with unfarnesylated peptides | Homo sapiens | KSKTKC(farnesyl) + VIM | - |
? |
Synonyms | Comment | Organism |
---|---|---|
human Ras-converting enzyme | abbrevation hRCE1 | Homo sapiens |