Application | Comment | Organism |
---|---|---|
medicine | most lethal biological substance have been weaponized in highly toxic aerosol form to pose a significant dual threat to both civilian and military populations, there is an urgent need for therapeutic countermeasures against BoNTs | Clostridium botulinum |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
amodiaquine | antimalarial drug, 30% inhibition | Clostridium botulinum | |
bisquinoline Q2-15 | 60% inhibition | Clostridium botulinum | |
bisquinoline Q2-61 | 50% inhibition | Clostridium botulinum | |
Chloroquine | antimalarial drug, 20% inhibition | Clostridium botulinum | |
NSC 119889 | 56% inhibition | Clostridium botulinum | |
NSC 130796 | 48% inhibition | Clostridium botulinum | |
NSC 357756 | 57% inhibition | Clostridium botulinum | |
NSC 402959 | 40% inhibition | Clostridium botulinum | |
NSC 625324 (silver sulfadiazine) | 100% inhibition | Clostridium botulinum | |
NSC 661755 (michellamine B) | 62% inhibition | Clostridium botulinum | |
NSC 86372 | 51% inhibition | Clostridium botulinum | |
Quinacrine | antimalarial drug, 30% inhibition | Clostridium botulinum |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
SNARE-protein + H2O | Clostridium botulinum | soluble NSF-attachment protein receptor | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Clostridium botulinum | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
SNAP-25 + H2O | - |
Clostridium botulinum | ? | - |
? | |
SNARE-protein + H2O | soluble NSF-attachment protein receptor | Clostridium botulinum | ? | - |
? | |
synaptobrevin + H2O | - |
Clostridium botulinum | ? | - |
? | |
Syntaxin + H2O | - |
Clostridium botulinum | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
BoNT | - |
Clostridium botulinum |
BoNT/A LC | - |
Clostridium botulinum |
neurotoxin A | - |
Clostridium botulinum |