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Literature summary for 3.4.24.15 extracted from

  • Molina, H.M.; Carmona, A.K.; Kouyoumdjian, M.; Borges, D.R.
    Thimet oligopeptidase EC 3.4.24.15 is a major liver kininase (2000), Life Sci., 67, 509-520.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
captopril 0.005 mM Rattus norvegicus
HVVR-4-nitroanilide
-
Rattus norvegicus
N-[1(R,S)-carboxy-3-phenylpropyl]-Ala-Ala-Phe-p-aminobenzoate 0.005 mM Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
liver
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
(o-aminobenzoyl)-Phe-Arg-Lys-(dinitrophenyl-proline) + H2O
-
Rattus norvegicus (o-aminobenzoyl)-Phe-Arg + Lys-(dinitrophenyl-proline)
-
?
(o-aminobenzoyl)-RPPGFSPFR-(N-(2,4-dinitrophenyl)ethylenediamine) + H2O
-
Rattus norvegicus (o-aminobenzoyl)-RPPGF + SPFR-(N-(2,4-dinitrophenyl)ethylenediamine)
-
?
(o-aminobenzoyl)-RPPGFSPFRQ-(N-(2,4-dinitrophenyl)ethylenediamine) + H2O
-
Rattus norvegicus (o-aminobenzoyl)-RPPGFSP + FRQ-(N-(2,4-dinitrophenyl)ethylenediamine)
-
?
N-succinyl-Gly-Pro-4-methylcoumaryl-7-amide + H2O
-
Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
BIE
-
Rattus norvegicus
bradykinin-inactivating endopeptidase
-
Rattus norvegicus