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Literature summary for 3.4.23.B8 extracted from

  • Akaji, K.; Teruya, K.; Aimoto, S.
    Solid-Phase Synthesis of HTLV-1 Protease Inhibitors Containing Hydroxyethylamine Dipeptide Isostere (2003), J. Org. Chem., 68, 4755-4763.
    View publication on PubMed
Search for more literature for 3.4.23.B8

Inhibitors

Inhibitors Comment Organism Structure
H-Pro-Val-Ile-hydroxyethylamine[(R)-isobutyl,(R)-hydroxy]-Pro-NH-CH2-C6H4I
-
 Human T-cell leukemia virus type I
H-Pro-Val-Ile-hydroxyethylamine[(R)-isobutyl,(S)-hydroxy]-Pro-NH-CH2-C6H4I
-
 Human T-cell leukemia virus type I
H-Pro-Val-Ile-hydroxyethylamine[(S)-isobutyl,(R)-hydroxy]-Pro-NH-CH2-C6H4I
-
 Human T-cell leukemia virus type I
H-Pro-Val-Ile-hydroxyethylamine[(S)-isobutyl,(S)-hydroxy]-Pro-NH-CH2-C6H4I
-
 Human T-cell leukemia virus type I

Organism

Organism UniProt Comment Textmining
Human T-cell leukemia virus type I
-
-
-

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.00494
-
 H-Pro-Val-Ile-hydroxyethylamine[(R)-isobutyl,(R)-hydroxy]-Pro-NH-CH2-C6H4I
-
 Human T-cell leukemia virus type I
0.00549
-
 H-Pro-Val-Ile-hydroxyethylamine[(S)-isobutyl,(S)-hydroxy]-Pro-NH-CH2-C6H4I
-
 Human T-cell leukemia virus type I
0.038
-
 H-Pro-Val-Ile-hydroxyethylamine[(S)-isobutyl,(R)-hydroxy]-Pro-NH-CH2-C6H4I
-
 Human T-cell leukemia virus type I
0.292
-
 H-Pro-Val-Ile-hydroxyethylamine[(R)-isobutyl,(S)-hydroxy]-Pro-NH-CH2-C6H4I
-
 Human T-cell leukemia virus type I