Inhibitors | Comment | Organism | Structure |
---|---|---|---|
diazoacetyl-norleucine methyl ester | - |
Cynara cardunculus | |
pepstatin | - |
Cynara cardunculus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.081 | - |
Leu-Ser-Phe(NO2)-Ahx-Ala-Leu-OMe | pH 4.7, 37°C | Cynara cardunculus | |
0.108 | - |
Lys-Pro-Ala-Glu-Phe-Phe-Phe(NO2)-Ala-Leu | pH 4.7, 37°C | Cynara cardunculus | |
0.11 | - |
Lys-Pro-Ala-Glu-Phe-Phe-Phe(NO2)-Ala-Leu | pH 4.7, 37°C | Cynara cardunculus | |
0.64 | - |
Leu-Ser-Phe(NO2)-Ahx-Ala-Leu-OMe | pH 4.7, 37°C | Cynara cardunculus |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
15000 | - |
x * 31000, and x * 15000, SDS-PAGE | Cynara cardunculus |
15000 | - |
x * 34000, and x * 15000, SDS-PAGE | Cynara cardunculus |
31000 | - |
x * 31000, and x * 15000, SDS-PAGE | Cynara cardunculus |
34000 | - |
x * 34000, and x * 15000, SDS-PAGE | Cynara cardunculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Cynara cardunculus | Q9XFX3 | isoform CardA | - |
Cynara cardunculus | Q9XFX4 | isoform CardB | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
91.8 | - |
pH 4.7, 37°C | Cynara cardunculus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Leu-Ser-Phe(NO2)-Ahx-Ala-Leu-OMe + H2O | - |
Cynara cardunculus | ? | - |
? | |
Leu-Ser-Phe(NO2)-Ahx-Ala-Leu-OMe + H2O | substrate of cardosin B | Cynara cardunculus | ? | - |
? | |
Lys-Pro-Ala-Glu-Phe-Phe-Phe(NO2)-Ala-Leu + H2O | - |
Cynara cardunculus | ? | - |
? | |
Lys-Pro-Ala-Glu-Phe-Phe-Phe(NO2)-Ala-Leu + H2O | substrate of cardosin A | Cynara cardunculus | ? | - |
? | |
Lys-Pro-Ala-Glu-Phe-Phe-Phe(NO2)-Ala-Leu + H2O | - |
Cynara cardunculus | Lys-Pro-Ala-Glu-Phe-Phe + Phe(NO2)-Ala-Leu + H2O | - |
? |
Subunits | Comment | Organism |
---|---|---|
? | x * 31000, and x * 15000, SDS-PAGE | Cynara cardunculus |
? | x * 34000, and x * 15000, SDS-PAGE | Cynara cardunculus |
Synonyms | Comment | Organism |
---|---|---|
CardA | - |
Cynara cardunculus |
cardB | - |
Cynara cardunculus |
Temperature Stability Minimum [°C] | Temperature Stability Maximum [°C] | Comment | Organism |
---|---|---|---|
60 | - |
stable up to | Cynara cardunculus |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
13.7 | - |
Leu-Ser-Phe(NO2)-Ahx-Ala-Leu-OMe | pH 4.7, 37°C | Cynara cardunculus | |
55.63 | - |
Lys-Pro-Ala-Glu-Phe-Phe-Phe(NO2)-Ala-Leu | pH 4.7, 37°C | Cynara cardunculus | |
86.2 | - |
Leu-Ser-Phe(NO2)-Ahx-Ala-Leu-OMe | pH 4.7, 37°C | Cynara cardunculus | |
89.4 | - |
Lys-Pro-Ala-Glu-Phe-Phe-Phe(NO2)-Ala-Leu | pH 4.7, 37°C | Cynara cardunculus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
5 | - |
- |
Cynara cardunculus |
pH Minimum | pH Maximum | Comment | Organism |
---|---|---|---|
2 | 7 | - |
Cynara cardunculus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000001 | - |
pepstatin | pH 4.7, 37°C | Cynara cardunculus | |
0.000003 | - |
pepstatin | pH 4.7, 37°C | Cynara cardunculus |
kcat/KM Value [1/mMs-1] | kcat/KM Value Maximum [1/mMs-1] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
21.3 | - |
Leu-Ser-Phe(NO2)-Ahx-Ala-Leu-OMe | pH 4.7, 37°C | Cynara cardunculus | |
515.1 | - |
Lys-Pro-Ala-Glu-Phe-Phe-Phe(NO2)-Ala-Leu | pH 4.7, 37°C | Cynara cardunculus | |
808.3 | - |
Lys-Pro-Ala-Glu-Phe-Phe-Phe(NO2)-Ala-Leu | pH 4.7, 37°C | Cynara cardunculus | |
1066 | - |
Leu-Ser-Phe(NO2)-Ahx-Ala-Leu-OMe | pH 4.7, 37°C | Cynara cardunculus |