Crystallization (Comment) | Organism |
---|---|
plasmepsin II in complex with pepstatin A | Plasmodium falciparum |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Ro40-4388 | - |
Plasmodium falciparum | |
Ro40-5576 | - |
Plasmodium falciparum |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Plasmodium falciparum | - |
- |
- |
Posttranslational Modification | Comment | Organism |
---|---|---|
proteolytic modification | recombinant proplasmepsin II autoactivates at acidic pH, but the location of the cleavage site varies dependening on the conditions used | Plasmodium falciparum |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00025 | - |
Ro40-5576 | - |
Plasmodium falciparum | |
0.0007 | - |
Ro40-4388 | - |
Plasmodium falciparum |