Crystallization (Comment) | Organism |
---|---|
vapour diffusion, space group P3(2)21, in complex with inhibitor CP-81,198 unit cell dimensions a : b : 86.8 A, c : 110.2 A, in complex with inhibitor CP-108,420 unit cell dimensions a : b : 86.9 A, c : 110.2 A, in complex with inhibitor CP-72,647 unit cell dimensions a : b : 86.4 A, c : 109.9 A, in complex with inhibitor PD-129,541 unit cell dimensions a : b : 87.3 A, c : 110.7 A, in complex with inhibitor PD-133,450 unit cell dimensions a : b : 86.9 A, c : 110.2 A | Saccharomyces cerevisiae |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
CP-108,420 | - |
Saccharomyces cerevisiae | |
CP-72,647 | - |
Saccharomyces cerevisiae | |
CP-81,198 | - |
Saccharomyces cerevisiae | |
CP-81,282 | - |
Saccharomyces cerevisiae | |
PD-129,541 | cyclic peptide inhibitor | Saccharomyces cerevisiae | |
PD-133,450 | - |
Saccharomyces cerevisiae |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
42000 | - |
- |
Saccharomyces cerevisiae |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Saccharomyces cerevisiae | - |
baker's yeast | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
haemoglobin + H2O | - |
Saccharomyces cerevisiae | ? | - |
? |
Subunits | Comment | Organism |
---|---|---|
monomer | - |
Saccharomyces cerevisiae |
Synonyms | Comment | Organism |
---|---|---|
Proteinase A | - |
Saccharomyces cerevisiae |
vacuolar aspartic proteinase | - |
Saccharomyces cerevisiae |
yeast proteinase | - |
Saccharomyces cerevisiae |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
3 | - |
for haemoglobin cleavage | Saccharomyces cerevisiae |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000004 | - |
PD-129,541 | pH 4.7, 37°C | Saccharomyces cerevisiae | |
0.0000071 | - |
CP-81,282 | pH 4.7, 37°C | Saccharomyces cerevisiae | |
0.0000137 | - |
PD-133,450 | pH 4.7, 37°C | Saccharomyces cerevisiae | |
0.000398 | - |
CP-108,420 | pH 4.7, 37°C | Saccharomyces cerevisiae | |
0.0009418 | - |
CP-81,198 | pH 4.7, 37°C | Saccharomyces cerevisiae | |
0.003742 | - |
CP-72,647 | pH 4.7, 37°C | Saccharomyces cerevisiae |