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Literature summary for 3.4.22.62 extracted from

  • Yun, C.Y.; Liu, S.; Lim, S.F.; Wang, T.; Chung, B.Y.; Jiat Teo, J.; Chuan, K.H.; Soon, A.S.; Goh, K.S.; Song, Z.
    Specific inhibition of caspase-8 and -9 in CHO cells enhances cell viability in batch and fed-batch cultures (2007), Metab. Eng., 9, 406-418.
    View publication on PubMed

Cloned(Commentary)

Cloned (Comment) Organism
expression in Escherichia coli Cricetulus griseus

Inhibitors

Inhibitors Comment Organism Structure
benzyloxycarbonyl-Ile-Glu-Thr-Asp-fluoromethylketone
-
Cricetulus griseus
benzyloxycarbonyl-Leu-Glu-His-Asp-fluoromethylketone
-
Cricetulus griseus
benzyloxycarbonyl-Val-Asp-Val-Ala-Asp-fluoromethylketone
-
Cricetulus griseus
additional information inhibition of caspase-9 enhances the viability of the CHO cells in both batch and fed-batch suspension cultures Cricetulus griseus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
additional information Cricetulus griseus caspase-9 is possibly involved in the apoptotic cell death in batch and fed-batch cultures of CHO cells ?
-
?

Organism

Organism UniProt Comment Textmining
Cricetulus griseus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
CHO cell inhibition of caspase-9 enhances the viability of the CHO cells in both batch and fed-batch suspension cultures. Caspase-9 is possible involved in the apoptotic cell death in batch and fed-batch cultures of CHO cells Cricetulus griseus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
acetyl-Ile-Glu-Thr-Asp-p-nitroanilide + H2O 13% of the activity with acetyl-Leu-Glu-His-Asp-p-nitroanilide Cricetulus griseus acetyl-Ile-Glu-Thr-Asp + p-nitroaniline
-
?
acetyl-Leu-Glu-His-Asp-p-nitroanilide + H2O
-
Cricetulus griseus acetyl-Leu-Glu-His-Asp + p-nitroaniline
-
?
acetyl-Trp-Glu-His-Asp-p-nitroanilide + H2O 49% of the activity with acetyl-Leu-Glu-His-Asp-p-nitroanilide Cricetulus griseus acetyl-Trp-Glu-His-Asp + p-nitroaniline
-
?
acetyl-Val-Glu-Ile-Asp-p-nitroanilide + H2O 19% of the activity with acetyl-Leu-Glu-His-Asp-p-nitroanilide Cricetulus griseus acetyl-Val-Glu-Ile-Asp + p-nitroaniline
-
?
additional information caspase-9 is possibly involved in the apoptotic cell death in batch and fed-batch cultures of CHO cells Cricetulus griseus ?
-
?
additional information no activity with acetyl-Asp-Glu-Val-Asp-p-nitroanilide and acetyl-Val-Asp-Val-Ala-Asp-p-nitroanilide Cricetulus griseus ?
-
?