Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 3.4.22.56 extracted from

  • Garcia-Calvo, M.; Peterson, E.P.; Leiting, B.; Ruel, R.; Nicholson, D.W.; Thornberry, N.A.
    Inhibition of human caspases by peptide-based and macromolecular inhibitors (1998), J. Biol. Chem., 273, 32608-32613.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
acetyl-AEVD-aldehyde
-
Homo sapiens
acetyl-DEVD-aldehyde
-
Homo sapiens
acetyl-IETD-aldehyde
-
Homo sapiens
acetyl-WEHD-aldehyde
-
Homo sapiens
benzyloxycarbonyl-Val-Ala-Asp-fluoromethylketone t1/2 at 0.001 mM is 43 s Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.00000023
-
acetyl-DEVD-aldehyde pH 7.5, 25°C Homo sapiens
0.000042
-
acetyl-AEVD-aldehyde pH 7.5, 25°C Homo sapiens
0.000195
-
acetyl-IETD-aldehyde pH 7.5, 25°C Homo sapiens
0.0016
-
cowpox serpin CrmA pH 7.5, 25°C Homo sapiens
0.00196
-
acetyl-WEHD-aldehyde pH 7.5, 25°C Homo sapiens