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Literature summary for 3.4.22.52 extracted from

  • Inomata, M.; Nomoto, M.; Hayashi, M.; Nakamura, M.; Imahori, K.; Kawashima, S.
    Comparison of low and high calcium requiring forms of the calcium-activated neutral protease (CANP) from rabbit skeletal muscle (1984), J. Biochem., 95, 1661-1670.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
antipain 0.01 mM, 80-90% inhibition Oryctolagus cuniculus
E-64c 0.01 mM, 80-90% inhibition Oryctolagus cuniculus
leupeptin 0.01 mM, 80-90% inhibition Oryctolagus cuniculus
pepstatin A 1 mM, 60-80% inhibition Oryctolagus cuniculus
TLCK 0.1 mM, 60-80% inhibition Oryctolagus cuniculus

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.0081
-
succinyl-casein pH 7.5, 25°C Oryctolagus cuniculus
2
-
succinyl-bovine serum albumin pH 7.5, 25°C Oryctolagus cuniculus
63
-
succinyl-protamine pH 7.5, 25°C Oryctolagus cuniculus
283.5
-
succinyl-insulin B pH 7.5, 25°C Oryctolagus cuniculus

Metals/Ions

Metals/Ions Comment Organism Structure
Ba2+ activates, Ka: 1.5 mM Oryctolagus cuniculus
Ca2+ Ka-value : 0.05 mM Oryctolagus cuniculus
Mn2+ slight activation Oryctolagus cuniculus
Sr2+ activates, Ka: 0.45 mM Oryctolagus cuniculus

Organism

Organism UniProt Comment Textmining
Oryctolagus cuniculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
skeletal muscle
-
Oryctolagus cuniculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
succinyl-bovine serum albumin + H2O
-
Oryctolagus cuniculus ?
-
?
succinyl-bovine-serum-albumin + H2O
-
Oryctolagus cuniculus ?
-
?
succinyl-casein + H2O
-
Oryctolagus cuniculus ?
-
?
succinyl-insulin B + H2O
-
Oryctolagus cuniculus ?
-
?
succinyl-protamine + H2O
-
Oryctolagus cuniculus ?
-
?

Temperature Stability [°C]

Temperature Stability Minimum [°C] Temperature Stability Maximum [°C] Comment Organism
60
-
10 min, 15% loss of activity Oryctolagus cuniculus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.3
-
-
Oryctolagus cuniculus