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Literature summary for 3.4.22.43 extracted from

  • Puzer, L.; Cotrin, S.S.; Alves, M.F.; Egborge, T.; Araujo, M.S.; Juliano, M.A.; Juliano, L.; Broemme, D.; Carmona, A.K.
    Comparative substrate specificity analysis of recombinant human cathepsin V and cathepsin L (2004), Arch. Biochem. Biophys., 430, 274-283.
    View publication on PubMed

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
additional information
-
additional information
-
Homo sapiens
0.0006
-
2-aminobenzoyl-KLRVSKQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
0.0006
-
2-aminobenzoyl-KLRSIKQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
0.0008
-
2-aminobenzoyl-KK-epsilon-amino-caproic acid-ELKLQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
0.0012
-
2-aminobenzoyl-KLRSSKQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
0.0016
-
2-aminobenzoyl-ALRSSKQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
0.0017
-
2-aminobenzoyl-EE-epsilon-amino-caproic acid-ELKLQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
0.002
-
2-aminobenzoyl-ELKLQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
2-aminobenzoyl-ALRSSKQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O best substrate Homo sapiens ?
-
?
2-aminobenzoyl-EE-epsilon-amino-caproic acid-ELKLQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O
-
Homo sapiens ?
-
?
2-aminobenzoyl-ELKLQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O
-
Homo sapiens ?
-
?
2-aminobenzoyl-KK-epsilon-amino-caproic acid-ELKLQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O
-
Homo sapiens ?
-
?
2-aminobenzoyl-KLRSIKQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O best substrate Homo sapiens 2-aminobenzoyl-KLR + SIKQ-N-(2,4-dinitrophenyl)ethylenediamine
-
?
2-aminobenzoyl-KLRSSKQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O
-
Homo sapiens ?
-
?
2-aminobenzoyl-KLRSXKQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O X is varied with diverse amino acids, highest activity with Ile, kinetics, detailed overview Homo sapiens 2-aminobenzoyl-KLR + SXKQ-N-(2,4-dinitrophenyl)ethylenediamine
-
?
2-aminobenzoyl-KLRVSKQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O
-
Homo sapiens ?
-
?
2-aminobenzoyl-KLRXSKQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O X is varied with diverse amino acids, highest activity with Val, kinetics, detailed overview Homo sapiens 2-aminobenzoyl-KLR + XSKQ-N-(2,4-dinitrophenyl)ethylenediamine
-
?
2-aminobenzoyl-KLXSSKQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O X is varied with diverse amino acids, highest activity with Arg, kinetics, detailed overview Homo sapiens 2-aminobenzoyl-KLX + SSKQ-N-(2,4-dinitrophenyl)ethylenediamine
-
?
2-aminobenzoyl-KXRSSKQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O X is varied with diverse amino acids, highest activity with Leu, kinetics, detailed overview Homo sapiens ?
-
?
2-aminobenzoyl-XLRSSKQ-N-(2,4-dinitrophenyl)ethylenediamine + H2O X is varied with diverse amino acids, highest activity with Ala, kinetics, detailed overview Homo sapiens ?
-
?
kininogen fragments + H2O kininogenase activity with high and low molecular weight kininogens Homo sapiens ? Lys-bradykinin is the major product ?
additional information substrate and cleavage site specificity of activated recombinant enzyme, comparison to cathepsin L, overview Homo sapiens ?
-
?

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
37
-
assay at Homo sapiens

Turnover Number [1/s]

Turnover Number Minimum [1/s] Turnover Number Maximum [1/s] Substrate Comment Organism Structure
additional information
-
additional information
-
Homo sapiens
0.6
-
2-aminobenzoyl-ELKLQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
0.9
-
2-aminobenzoyl-KLRVSKQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
1.3
-
2-aminobenzoyl-KLRSSKQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
1.3
-
2-aminobenzoyl-EE-epsilon-amino-caproic acid-ELKLQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
1.5
-
2-aminobenzoyl-KLRSIKQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
1.7
-
2-aminobenzoyl-KK-epsilon-amino-caproic acid-ELKLQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens
4
-
2-aminobenzoyl-ALRSSKQ-N-(2,4-dinitrophenyl)ethylenediamine recombinant enzyme, pH 5.5, 37°C Homo sapiens

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
5.5 6.5 assay at Homo sapiens