Inhibitors | Comment | Organism | Structure |
---|---|---|---|
E64 | 64 nM | Homo sapiens | |
leupeptin | 5.2 nM | Homo sapiens | |
paecilopeptin | i.e. acetyl-Leu-Val-CHO, IC50: 21 nM | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
benzyloxycarbonyl-Val-Val-Arg-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | benzyloxycarbonyl-Val-Val-Arg + 7-amino-4-methylcoumarin | - |
? |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.000021 | - |
i.e. acetyl-Leu-Val-CHO, IC50: 21 nM | Homo sapiens | paecilopeptin |