Protein Variants | Comment | Organism |
---|---|---|
V133A/S205E | change in specificity compared to wild-type enzyme | Carica papaya |
V133A/V157G/S205E | important decrease in activity, change in specificity compared to the wild-type enzyme | Carica papaya |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.089 | - |
benzyloxycarbonyl-Phe-Arg 4-methylcoumarin-7-amide | - |
Carica papaya | |
0.191 | - |
benzyloxycarbonyl-Phe-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/S205E | Carica papaya | |
0.43 | - |
benzyloxycarbonyl-Phe-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/V157G/S205E | Carica papaya | |
0.94 | - |
benzyloxycarbonyl-Arg-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/S205E | Carica papaya | |
1.296 | - |
benzyloxycarbonyl-citrullyl-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/S205E | Carica papaya | |
1.48 | - |
benzyloxycarbonyl-Phe-Arg 4-methylcoumarin-7-amide | - |
Carica papaya | |
2.03 | - |
benzyloxycarbonyl-citrullyl-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/V157G/S205E | Carica papaya | |
2.27 | - |
benzyloxycarbonyl-Arg-Arg 4-methylcoumarin-7-amide | - |
Carica papaya | |
5.6 | - |
benzyloxycarbonyl-Arg-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/V157G/S205E | Carica papaya |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Carica papaya | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
benzyloxycarbonyl-Arg-Arg 4-methylcoumarin-7-amide + H2O | - |
Carica papaya | ? | - |
? | |
benzyloxycarbonyl-citrullyl-Arg 4-methylcoumarin-7-amide + H2O | - |
Carica papaya | ? | - |
? | |
benzyloxycarbonyl-Phe-Arg 4-methylcoumarin-7-amide + H2O | - |
Carica papaya | ? | - |
? |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.42 | - |
benzyloxycarbonyl-citrullyl-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/V157G/S205E | Carica papaya | |
0.79 | - |
benzyloxycarbonyl-Arg-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/V157G/S205E | Carica papaya | |
1.18 | - |
benzyloxycarbonyl-Arg-Arg 4-methylcoumarin-7-amide | - |
Carica papaya | |
2.78 | - |
benzyloxycarbonyl-Phe-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/V157G/S205E | Carica papaya | |
5.67 | - |
benzyloxycarbonyl-citrullyl-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/S205E | Carica papaya | |
8.14 | - |
benzyloxycarbonyl-citrullyl-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/V157G/S205E | Carica papaya | |
9.3 | - |
benzyloxycarbonyl-Arg-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/S205E | Carica papaya | |
16.9 | - |
benzyloxycarbonyl-Phe-Arg 4-methylcoumarin-7-amide | mutant enzyme V133A/S205E | Carica papaya | |
41.6 | - |
benzyloxycarbonyl-Phe-Arg 4-methylcoumarin-7-amide | - |
Carica papaya |