Inhibitors | Comment | Organism | Structure |
---|---|---|---|
amidinophenylmethansulfonylfluorid | complete inhibition at 2.5 microM | Homo sapiens | |
Aprotinin | 30% inhibition at 2.5 mM | Homo sapiens | |
benzamidine | 40% inhibition at 2.5 mM | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.27 | - |
Gln-Ala-Arg-7-amido-4-methylcoumarin | 20 mM Tris, 150 mM NaCl, 0.01% Tween 20, pH 7.5, 37°C | Homo sapiens | |
0.28 | - |
Val-Pro-Arg-7-amido-4-methylcoumarin | 20 mM Tris, 150 mM NaCl, 0.01% Tween 20, pH 7.5, 37°C | Homo sapiens | |
0.44 | - |
Phe-Ser-Arg-7-amido-4-methylcoumarin | 20 mM Tris, 150 mM NaCl, 0.01% Tween 20, pH 7.5, 37°C | Homo sapiens | |
0.53 | - |
Pro-Phe-Arg-7-amido-4-methylcoumarin | 20 mM Tris, 150 mM NaCl, 0.01% Tween 20, pH 7.5, 37°C | Homo sapiens | |
1.18 | - |
Gly-Pro-Arg-7-amido-4-methylcoumarin | 20 mM Tris, 150 mM NaCl, 0.01% Tween 20, pH 7.5, 37°C | Homo sapiens |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
40000 | - |
SDS-PAGE | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | Q9UBX7 | - |
- |
Purification (Comment) | Organism |
---|---|
to homogeneity by immunoaffinity chromatography and high-performance liquid chromatography | Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
seminal plasma | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Gln-Ala-Arg-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | Gln-Ala-Arg + 7-amino-4-methylcoumarin | - |
? | |
Gly-Pro-Arg-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | Gly-Pro-Arg + 7-amino-4-methylcoumarin | - |
? | |
Phe-Ser-Arg-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | Phe-Ser-Arg + 7-amino-4-methylcoumarin | - |
? | |
Pro-Phe-Arg-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | Pro-Phe-Arg + 7-amino-4-methylcoumarin | - |
? | |
Val-Pro-Arg-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | Val-Pro-Arg + 7-amino-4-methylcoumarin | - |
? |
Subunits | Comment | Organism |
---|---|---|
monomer | SDS-PAGE | Homo sapiens |
Synonyms | Comment | Organism |
---|---|---|
hK11 | - |
Homo sapiens |
human kallikrein 11 | - |
Homo sapiens |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.21 | - |
Gly-Pro-Arg-7-amido-4-methylcoumarin | 20 mM Tris, 150 mM NaCl, 0.01% Tween 20 (pH7.5), 37°C | Homo sapiens | |
0.23 | - |
Gln-Ala-Arg-7-amido-4-methylcoumarin | 20 mM Tris, 150 mM NaCl, 0.01% Tween 20 (pH7.5), 37°C | Homo sapiens | |
0.39 | - |
Phe-Ser-Arg-7-amido-4-methylcoumarin | 20 mM Tris, 150 mM NaCl, 0.01% Tween 20 (pH7.5), 37°C | Homo sapiens | |
0.45 | - |
Val-Pro-Arg-7-amido-4-methylcoumarin | 20 mM Tris, 150 mM NaCl, 0.01% Tween 20 (pH7.5), 37°C | Homo sapiens | |
1.86 | - |
Pro-Phe-Arg-7-amido-4-methylcoumarin | 20 mM Tris, 150 mM NaCl, 0.01% Tween 20 (pH7.5), 37°C | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.5 | - |
- |
Homo sapiens |