Protein Variants | Comment | Organism |
---|---|---|
I99A | substrate acetyl-IEPD-7-amino-4-methylcoumarin, drastic reduction in ratio kcat/Km | Rattus norvegicus |
I99A/N218A | 6fold increase in Km-value, substrate acetyl-IEFD-7-amino-4-methylcoumarin | Rattus norvegicus |
I99F | substrate acetyl-IEPD-7-amino-4-methylcoumarin, 6fold reduction in ratio kcat/Km | Rattus norvegicus |
I99R | substrate acetyl-IEPD-7-amino-4-methylcoumarin, 10fold reduction in ratio kcat/Km | Rattus norvegicus |
N218A | substrate acetyl-IEPD-7-amino-4-methylcoumarin, 30% reduction in ratio kcat/Km | Rattus norvegicus |
N218A/R192A | substrate acetyl-IEPD-7-amino-4-methylcoumarin, drastic reduction in ratio kcat/Km | Rattus norvegicus |
N218A/R192E | substrate acetyl-IEPD-7-amino-4-methylcoumarin, drastic reduction in ratio kcat/Km | Rattus norvegicus |
N218T | substrate acetyl-IEPD-7-amino-4-methylcoumarin, almost 2fold increase in ratio kcat/Km | Rattus norvegicus |
Y174A | substrate acetyl-IEPD-7-amino-4-methylcoumarin, 6fold reduction in ratio kcat/Km | Rattus norvegicus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.15 | - |
acetyl-IEFD-7-amido-4-methylcoumarin | wild-type | Rattus norvegicus | |
0.25 | - |
acetyl-IETD-4-methylcoumarin-7-amide | wild-type | Rattus norvegicus | |
0.37 | - |
acetyl-IEPD-7-amido-4-methylcoumarin | wild-type | Rattus norvegicus | |
0.6 | - |
acetyl-LEFD-7-amido-4-methylcoumarin | wild-type | Rattus norvegicus | |
0.88 | - |
acetyl-IEFD-7-amido-4-methylcoumarin | mutant I99A | Rattus norvegicus | |
0.89 | - |
acetyl-IEFD-7-amido-4-methylcoumarin | mutant I99A/N218A | Rattus norvegicus | |
0.93 | - |
acetyl-IEFD-7-amido-4-methylcoumarin | mutant I99R | Rattus norvegicus | |
1.1 | - |
acetyl-LEPD-7-amido-4-methylcoumarin | wild-type | Rattus norvegicus | |
1.18 | - |
acetyl-IKPD-7-amido-4-methylcoumarin | mutant N218T | Rattus norvegicus | |
1.3 | - |
acetyl-IEFD-7-amido-4-methylcoumarin | mutant I99A/N218A | Rattus norvegicus | |
1.6 | - |
acetyl-IKPD-7-amido-4-methylcoumarin | wild-type | Rattus norvegicus | |
1.8 | - |
acetyl-IKPD-7-amido-4-methylcoumarin | mutant N218A | Rattus norvegicus | |
2.7 | - |
acetyl-IEPD-7-amido-4-methylcoumarin | mutant I99A/N218A | Rattus norvegicus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | P18291 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
acetyl-IAPD-7-amido-4-methylcoumarin + H2O | - |
Rattus norvegicus | acetyl-IAPD + 7-amino-4-methylcoumarin | - |
? | |
acetyl-IEFD-7-amido-4-methylcoumarin + H2O | - |
Rattus norvegicus | acetyl-IEFD + 7-amino-4-methylcoumarin | - |
? | |
acetyl-IEPD-7-amido-4-methylcoumarin + H2O | - |
Rattus norvegicus | acetyl-IEPD + 7-amino-4-methylcoumarin | - |
? | |
acetyl-IETD-7-amido-4-methylcoumarin + H2O | - |
Rattus norvegicus | acetyl-IETD + 7-amino-4-methylcoumarin | - |
? | |
acetyl-IKPD-7-amido-4-methylcoumarin + H2O | - |
Rattus norvegicus | acetyl-IKPD + 7-amino-4-methylcoumarin | - |
? | |
acetyl-LEFD-7-amido-4-methylcoumarin + H2O | - |
Rattus norvegicus | acetyl-LEFD + 7-amino-4-methylcoumarin | - |
? | |
acetyl-LEPD-7-amido-4-methylcoumarin + H2O | - |
Rattus norvegicus | acetyl-LEPD + 7-amino-4-methylcoumarin | - |
? |
Synonyms | Comment | Organism |
---|---|---|
natural killer cell protease 1 | - |
Rattus norvegicus |