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Literature summary for 3.4.21.75 extracted from

  • Hatsuzawa, K.; Murakami, K.; Nakayama, K.
    Molecular and enzymatic properties of furin, a Kex2-like endoprotease involved in precursor cleavage at Arg-X-Lys/Arg-Arg sites (1992), J. Biochem., 111, 296-301.
    View publication on PubMed

Cloned(Commentary)

Cloned (Comment) Organism
-
Mus musculus

Inhibitors

Inhibitors Comment Organism Structure
antipain moderately Mus musculus
Cu2+
-
Mus musculus
diisopropyl fluorophosphate
-
Mus musculus
EDTA
-
Mus musculus
Hg2+
-
Mus musculus
leupeptin moderately Mus musculus
NEM moderately Mus musculus
p-chloromercuribenzenesulfonic acid
-
Mus musculus
Zn2+
-
Mus musculus

Localization

Localization Comment Organism GeneOntology No. Textmining
Golgi trans-face human, mainly, the enzyme can translocate between the cell surface and the trans-Golgi network Mus musculus
-
-

Metals/Ions

Metals/Ions Comment Organism Structure
Ca2+ required Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
-
expression in Chinese hamster ovary cells
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
Prorenin + H2O
-
Mus musculus ?
-
?
Protein precursor + H2O
-
Mus musculus ?
-
?
tert-butoxycarbonyl-Arg-Val-Arg-Arg-4-methylcoumarin 7-amide + H2O
-
Mus musculus tert-butoxycarbonyl-Arg-Val-Arg-Arg + 7-amino-4-methylcoumarin
-
?

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
6.5 7.5 tert-butoxycarbonyl-Arg-Val-Arg-Arg-4-methylcoumarin 7-amide Mus musculus
7
-
around, tert-butoxycarbonyl-Arg-Val-Arg-Arg-4-methylcoumarin 7-amide Mus musculus