Activating Compound | Comment | Organism | Structure |
---|---|---|---|
certoparin | clinical LMWH enhances activity | Homo sapiens | |
dalteparin | clinical LMWH enhances activity | Homo sapiens | |
dermatan sulfate | shows potent APC enhancing effect | Homo sapiens | |
enoxaparin | clinical LMWH enhances activity | Homo sapiens | |
glycosaminoglycan | enhances activity with factor V but not with factor Va as substrate | Homo sapiens | |
LMW heparin | enhances the anticoagulant action of activated protein C | Homo sapiens | |
nadroparin | clinical LMWH enhances activity | Homo sapiens | |
tinzaparin | clinical LMWH enhances activity | Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
factor V + H2O | Homo sapiens | proteolytic inactivation | ? | - |
? | |
factor VIII + H2O | Homo sapiens | proteolytic inactivation | ? | - |
? | |
Factor VIIIa + H2O | Homo sapiens | #> | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
human | - |
Purification (Comment) | Organism |
---|---|
- |
Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
factor V + H2O | proteolytic inactivation | Homo sapiens | ? | - |
? | |
factor VIII + H2O | proteolytic inactivation | Homo sapiens | ? | - |
? | |
Factor VIIIa + H2O | proteolytic inactivation | Homo sapiens | ? | - |
? | |
Factor VIIIa + H2O | #> | Homo sapiens | ? | - |
? |
Cofactor | Comment | Organism | Structure |
---|---|---|---|
chondroitin sulfate | anticoagulant cofactor for APC | Homo sapiens | |
dermatan sulfate | anticoagulant cofactor for APC, important physiological cofactor | Homo sapiens | |
heparan sulfate | anticoagulant cofactor for APC | Homo sapiens |