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Literature summary for 3.4.21.68 extracted from

  • Komissarov, A.A.; Declerck, P.J.; Shore, J.D.
    Protonation State of a Single Histidine Residue Contributes Significantly to the Kinetics of the Reaction of Plasminogen Activator Inhibitor-1 with Tissue-type Plasminogen Activator (2004), J. Biol. Chem., 279, 23007-23013.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
N-((2-(iodoacetoxy)ethyl)-N-methyl)amino-7-nitrobenz-2-oxa-3-diazole P9 plasminogen activator inhibitor-1 Homo sapiens

Molecular Weight [Da]

Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
63500
-
x * 63500, SDS-PAGE Homo sapiens

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
plasminogen + H2O Homo sapiens
-
plasmin + ?
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens P00750
-
-

Source Tissue

Source Tissue Comment Organism Textmining

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
plasminogen + H2O
-
Homo sapiens plasmin + ?
-
?

Subunits

Subunits Comment Organism
? x * 63500, SDS-PAGE Homo sapiens

Synonyms

Synonyms Comment Organism
Tissue-type plasminogen activator
-
Homo sapiens
tPA
-
Homo sapiens