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Literature summary for 3.4.21.59 extracted from

  • Mori, S.; Itoh, Y.; Shinohata, R.; Sendo, T.; Oishi, R.; Nishibori, M.
    Nafamostat mesilate is an extremely potent inhibitor of human tryptase (2003), J. Pharm. Sci., 92, 420-423.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
6-amidino-2-naphthyl p-guanidinobenzoate dimethane sulfonate nafamostat mesilate Homo sapiens
gabexate mesilate
-
Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
human
-

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.0000000953
-
6-amidino-2-naphthyl p-guanidinobenzoate dimethane sulfonate pH 7.8, 37°C Homo sapiens
0.0000951
-
gabexate mesilate pH 7.8, 37°C Homo sapiens