Protein Variants | Comment | Organism |
---|---|---|
R463X | the mutations Arg463Gln, Arg463Lys or Arg463Phe all stabilize the zymogen state | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
diisopropyl fluorophosphate | - |
Homo sapiens | |
additional information | above 0.0005 mM C1rbar the enzyme aggregates with loss of activity | Homo sapiens | |
p-amidinophenylmethylsulfonyl fluoride | - |
Homo sapiens | |
p-tosyl-Lys-chloromethyl ketone | - |
Homo sapiens | |
phenylmethylsulfonyl fluoride | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
N-acetyl-Arg methyl ester + H2O | - |
Homo sapiens | N-acetyl-Arg + methanol | - |
? | |
N-acetyl-Gly-Lys methyl ester + H2O | - |
Homo sapiens | N-acetyl-Gly-Lys + methanol | - |
? | |
N-carbobenzoxy-Lys-p-nitrophenyl ester + H2O | - |
Homo sapiens | N-carbobenzoxy-Lys + 4-nitrophenyl | - |
? | |
N-carbobenzoxy-Tyr-p-nitrophenyl ester + H2O | - |
Homo sapiens | N-carbobenzoxy-Tyr + 4-nitrophenol | - |
? |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
12.5 | - |
N-Acetyl-Gly-Lys methyl ester | - |
Homo sapiens | |
18.3 | - |
N-acetyl-Arg methyl ester | - |
Homo sapiens |