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Literature summary for 3.4.21.39 extracted from

  • Woodward, S.L.; Fraser, S.A.; Winkler, U.; Jackson, D.S.; Kam, C.M.; Powers, J.C.; Hudig, D.
    Purification and characterization of lymphocyte chymase I, a granzyme implicated in perforin-mediated lysis (1998), J. Immunol., 160, 4988-1993.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
2-(benzyloxycarbonyl-NH(CH2)2CONH)C6H4SO2F
-
Rattus norvegicus
3,4-dichloroisocoumarin
-
Rattus norvegicus
5-fluoresceinylthiocarbamoyl-Ala-Ala-Met phosphonate diphenyl ester
-
Rattus norvegicus
benzyloxycarbonyl-Gly-Leu-Phe-chloromethyl ketone
-
Rattus norvegicus
biotinyl-6-aminocaproyl-6-aminocaproyl-Phe-Leu-Phe-phosphonate phenyl ester
-
Rattus norvegicus
phenylmethylsulfonyl fluoride
-
Rattus norvegicus
succinyl-Phe-Leu-Phe-phosphonate diphenyl ester
-
Rattus norvegicus
tosyl-Phe-CH2Cl
-
Rattus norvegicus

Localization

Localization Comment Organism GeneOntology No. Textmining
specific granule rat natural killer cell (RNK)-16 granules Rattus norvegicus 42581
-

Molecular Weight [Da]

Molecular Weight [Da] Molecular Weight Maximum [Da] Comment Organism
30000
-
x * 30000, SDS-PAGE Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Rattus norvegicus

Source Tissue

Source Tissue Comment Organism Textmining
lymphocyte
-
Rattus norvegicus
-
mast cell
-
Rattus norvegicus
-
natural killer cell
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
additional information the enzyme from lymphocytes has a substrate preference for tryptophan, a preference distinct from rat mast cell chymase Rattus norvegicus ?
-
?
succinyl-Phe-Leu-Phe-thiobenzyl ester + H2O
-
Rattus norvegicus ?
-
?
t-butyloxycarbonyl-Ala-Ala-Asp-thiobenzyl ester + H2O
-
Rattus norvegicus ?
-
?
t-butyloxycarbonyl-Ala-Ala-Leu-thiobenzyl ester + H2O
-
Rattus norvegicus ?
-
?
t-butyloxycarbonyl-Ala-Ala-Met-thiobenzyl ester + H2O
-
Rattus norvegicus ?
-
?
t-butyloxycarbonyl-Ala-Ala-Phe-thiobenzyl ester + H2O
-
Rattus norvegicus ?
-
?
t-butyloxycarbonyl-Ala-Ala-Ser-thiobenzyl ester + H2O weak activity Rattus norvegicus ?
-
?
t-butyloxycarbonyl-Ala-Ala-Trp-thiobenzyl ester + H2O
-
Rattus norvegicus ?
-
?

Subunits

Subunits Comment Organism
? x * 30000, SDS-PAGE Rattus norvegicus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.5 9
-
Rattus norvegicus