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Literature summary for 3.4.21.37 extracted from

  • Hagio, T.; Kishikawa, K.; Kawabata, K.; Tasaka, S.; Hashimoto, S.; Hasegawa, N.; Ishizaka, A.
    Inhibition of neutrophil elastase reduces lung injury and bacterial count in hamsters (2008), Pulm. Pharmacol. Ther., 21, 884-891.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
sivelestat i.e. N-[2-[4-(2,2-dimethyl-propionyloxy)phenylsulfonylamino]benzoyl]aminoacetatetetrahydrate or ONO-5046, specific neutrophil elastase inhibitor, intravenous infusion of sivelestat at 3 mg/kg/h 0-22 h after Streptococcus pneumoniae inoculation reduces the increase in neutrophil elastase activity Mesocricetus auratus

Organism

Organism UniProt Comment Textmining
Mesocricetus auratus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
bronchoalveolar lavage fluid
-
Mesocricetus auratus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
N-methoxysuccinyl-Ala-Ala-Pro-Val-4-nitroanilide + H2O highly specific synthetic substrate for neutrophil elastase Mesocricetus auratus N-methoxysuccinyl-Ala-Ala-Pro-Val + 4-nitroaniline
-
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Synonyms

Synonyms Comment Organism
neutrophil elastase
-
Mesocricetus auratus