Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 3.4.21.27 extracted from

  • Pedicord, D.L.; Seiffert, D.; Blat, Y.
    Substrate-dependent modulation of the mechanism of factor XIa inhibition (2004), Biochemistry, 43, 11883-11888.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
Aprotinin
-
Homo sapiens
leupeptin
-
Homo sapiens

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
0.151
-
factor IX at 22°C Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
factor IX + H2O FIX Homo sapiens factor IXa + ?
-
?
L-pyroglutamyl-L-prolyl-L-arginyl-p-nitroanilide + H2O
-
Homo sapiens L-pyroglutamyl-L-prolyl-L-arginine + p-nitroaniline
-
?

Synonyms

Synonyms Comment Organism
factor XIa
-
Homo sapiens
FXIa
-
Homo sapiens

Turnover Number [1/s]

Turnover Number Minimum [1/s] Turnover Number Maximum [1/s] Substrate Comment Organism Structure
0.66
-
factor IX at 22°C Homo sapiens

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.52
-
Aprotinin L-pyroglutamyl-L-prolyl-L-arginyl-p-nitroanilide substrate, free FXIa Homo sapiens
0.96
-
Aprotinin FIX substrate, free FXIa Homo sapiens
1.43
-
leupeptin L-pyroglutamyl-L-prolyl-L-arginyl-p-nitroanilide substrate, free FXIa Homo sapiens
2.91
-
leupeptin FIX substrate, free FXIa Homo sapiens
10.42
-
Aprotinin FIX substrate, FXIa-FIX complex Homo sapiens
19.12
-
leupeptin FIX substrate, FXIa-FIX complex Homo sapiens
209
-
leupeptin L-pyroglutamyl-L-prolyl-L-arginyl-p-nitroanilide substrate, FXIa-FIX complex Homo sapiens