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Literature summary for 3.4.19.6 extracted from

  • Cruz, R.; Vargas, M.A.; Uribe, R.M.; Pascual, I.; Lazcano, I.; Yiotakis, A.; Matziari, M.; Joseph-Bravo, P.; Charli, J.L.
    Anterior pituitary pyroglutamyl peptidase II activity controls TRH-induced prolactin release (2008), Peptides, 29, 1953-1964.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
Glp-PSI[P(O)(OH)CH2]-His-Pro-NH2 phosphinic analogue of thyrotropin releasing hormone Rattus norvegicus
Hermodice carunculata peptidase inhibitor HcPI Rattus norvegicus

Localization

Localization Comment Organism GeneOntology No. Textmining
membrane
-
Rattus norvegicus 16020
-

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
thyrotropin releasing hormone + H2O Rattus norvegicus
-
?
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
female wistar rat
-

Source Tissue

Source Tissue Comment Organism Textmining
anterior pituitary
-
Rattus norvegicus
-
pituitary gland cell line
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
additional information hydrolyzing of substrates with the general structure pGlu-X-Y, X being a moderately bulky and uncharged residue and Y, either Pro, Ala, Trp, Pro-Gly, ProNH2, Pro-beta-naphthylamine, or Pro-7-amino-4-methyl coumarin Rattus norvegicus ?
-
?
thyrotropin releasing hormone + H2O
-
Rattus norvegicus ?
-
?
thyrotropin releasing hormone-beta-naphthylamine + H2O substrate activity assay Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
PPII
-
Rattus norvegicus
pyroglutamyl peptidase II
-
Rattus norvegicus

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
37
-
activity assay Rattus norvegicus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.5
-
activity assay Rattus norvegicus