Literature summary for 3.4.16.2 extracted from

Moreira, C.R.; Schmaier, A.H.; Mahdi, F.; da Motta, G.; Nader, H.B.; Shariat-Madar, Z.
Identification of prolylcarboxypeptidase as the cell matrix-associated prekallikrein activator (2002), FEBS Lett., 523, 167-170.

Search for more literature for 3.4.16.2

Inhibitors

Inhibitors	Comment	Organism	Structure
angiotensin II	IC50: 0.1 mM	Homo sapiens
antipain	IC50: 0.05 mM	Homo sapiens
bradykinin	IC50: 3 mM	Homo sapiens
corn trypsin inhibitor	IC50: 100 nM	Homo sapiens
N-(9-fluorenyl)methoxycarbonyl-aminoacylpyrrolidine-2-nitrile	IC50: 0.1 mM	Homo sapiens

Organism

Organism	UniProt	Comment	Textmining
Homo sapiens	-	-	-

Source Tissue

Source Tissue	Comment	Organism	Textmining
umbilical vein endothelial cell line	matrix	Homo sapiens	-

Synonyms

Synonyms	Comment	Organism
matrix PK activator	-	Homo sapiens

IC50 Value

IC50 Value	IC50 Value Maximum	Comment	Organism	Inhibitor	Structure
0.0001	-	IC50: 100 nM	Homo sapiens	corn trypsin inhibitor
0.05	-	IC50: 0.05 mM	Homo sapiens	antipain
0.1	-	IC50: 0.1 mM	Homo sapiens	angiotensin II
0.1	-	IC50: 0.1 mM	Homo sapiens	N-(9-fluorenyl)methoxycarbonyl-aminoacylpyrrolidine-2-nitrile
3	-	IC50: 3 mM	Homo sapiens	bradykinin

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Release 2023.1 (January 2023)