Inhibitors | Comment | Organism | Structure |
---|---|---|---|
alogliptin | - |
Homo sapiens | |
linagliptin | - |
Homo sapiens | |
saxagliptin | highly selective dipeptidyl peptidase-IV inhibitor for the treatment of type 2 diabetes, synonyms are BMS-477118, Onglyza, and saxagliptin hydrate, saxagliptin is 400fold and 75fold more potent against DPP-IV than DPP-8 or DPP-9 respectively, DPP-IV is inhibited dose-dependently, with maximal inhibition at 150 mg/day | Homo sapiens | |
sitagliptin | - |
Homo sapiens | |
vildagliptin | - |
Homo sapiens |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
glucagon-like peptide 1 + H2O | Homo sapiens | - |
? | - |
? | |
glucose-dependent insulinotropic peptide + H2O | Homo sapiens | - |
? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
blood plasma | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
glucagon-like peptide 1 + H2O | - |
Homo sapiens | ? | - |
? | |
glucose-dependent insulinotropic peptide + H2O | - |
Homo sapiens | ? | - |
? | |
Gly-L-Pro-4-nitroanilide | - |
Homo sapiens | Gly-L-Pro + 4-nitroaniline | - |
? | |
Gly-L-Pro-7-amido-4-methylcoumarin + H2O | - |
Homo sapiens | Gly-L-Pro + 7-amino-4-methylcoumarin | - |
? |
Synonyms | Comment | Organism |
---|---|---|
dipeptidyl peptidase-IV | - |
Homo sapiens |
DPP-IV | - |
Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0000006 | - |
saxagliptin | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00003 | - |
- |
Homo sapiens | saxagliptin |