Inhibitors | Comment | Organism | Structure |
---|---|---|---|
bestatin | Ki: 0.004 mM | Rattus norvegicus | |
EDTA | 60-80% inhibition at 20 mM | Rattus norvegicus | |
puromycin | Ki: 0.1 mM, low sensitivity to puromycin | Rattus norvegicus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.02 | - |
Leu-2-naphthylamide | from brain | Rattus norvegicus | |
0.025 | - |
L-Arg-2-naphthylamide | from kidney | Rattus norvegicus | |
0.027 | - |
L-Arg-2-naphthylamide | from brain | Rattus norvegicus | |
0.027 | - |
Leu-2-naphthylamide | from kidney | Rattus norvegicus | |
0.038 | - |
Ala-2-naphthylamide | from kidney | Rattus norvegicus | |
0.04 | - |
Ala-2-naphthylamide | from brain | Rattus norvegicus | |
0.045 | - |
Leu5-enkephalin | from brain | Rattus norvegicus | |
0.045 | - |
Met5-enkephalin | from brain | Rattus norvegicus | |
0.06 | - |
Met5-enkephalin | from kidney | Rattus norvegicus | |
0.065 | - |
Leu5-enkephalin | from kidney | Rattus norvegicus | |
0.8 | - |
Gly-2-naphthylamide | from brain | Rattus norvegicus | |
1 | - |
Gly-2-naphthylamide | from kidney | Rattus norvegicus | |
2.1 | 2.9 | Phe-Gly | - |
Rattus norvegicus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
membrane | cerebral membrane | Rattus norvegicus | 16020 | - |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Cd2+ | reactivation after inhibition by EDTA | Rattus norvegicus | |
Co2+ | reactivation after inhibition by EDTA | Rattus norvegicus | |
Mn2+ | reactivation after inhibition by EDTA | Rattus norvegicus | |
Zn2+ | reactivation after inhibition by EDTA | Rattus norvegicus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
aminoacyl peptide | Rattus norvegicus | - |
? | - |
? | |
enkephalin | Rattus norvegicus | may be involved in enkephalin neurotransmitter inactivation | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Rattus norvegicus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | - |
Rattus norvegicus | - |
kidney | - |
Rattus norvegicus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
aminoacyl peptide | - |
Rattus norvegicus | ? | - |
? | |
aminoacyl-2-naphthylamide + H2O | - |
Rattus norvegicus | amino acid + 2-naphthylamine | - |
? | |
enkephalin | may be involved in enkephalin neurotransmitter inactivation | Rattus norvegicus | ? | - |
? | |
Gly-2-naphthylamide + H2O | - |
Rattus norvegicus | Gly + 2-naphthylamine | - |
? | |
L-Arg-2-naphthylamide + H2O | - |
Rattus norvegicus | L-Arg + 2-naphthylamine | - |
? | |
Leu-2-naphthylamide + H2O | - |
Rattus norvegicus | Leu + 2-naphthylamine | - |
? | |
Leu5-enkephalin + H2O | - |
Rattus norvegicus | tyrosin + (2-5)Leu5-enkephalin | - |
? | |
Met5-enkephalin + H2O | - |
Rattus norvegicus | tyrosin + (2-5)Met5-enkephalin | - |
? | |
Phe-Gly + H2O | - |
Rattus norvegicus | Phe + Gly | - |
? |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.004 | - |
bestatin | - |
Rattus norvegicus |