Inhibitors | Comment | Organism | Structure |
---|---|---|---|
additional information | the PG500 series of heparan sulfate mimetics potently block the enzymatic activity of heparanase (fully sulfated, single entity oligosaccharides attached to a lipophilic moiety, which have been optimized for drug development) | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | Q9Y251 | - |
- |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | PG517: 162 nM, PG518: 59 nM, PG536: 6 nM, PG537: 6 nM, PG545: 6 nM, PG546: 4 nM, PG547: 16 nM, PG554: 9 nM, PG561: 11 nM, PG562: 9 nM, PI-88: 8 nM | Homo sapiens |