Cloned (Comment) | Organism |
---|---|
Epac1-camps-PDE4A1 fusion protein is expressed in HEK-293 cells | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
3-isobuytl-1-methylxanthine | - |
Homo sapiens | |
Ro20-1724 | PDE4 inhibitor | Homo sapiens | |
rolipram | PDE4 inhibitor | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P27815 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
3',5'-cAMP + H2O | - |
Homo sapiens | 5'-AMP | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PDE4 | - |
Homo sapiens |
PDE4A1 | isoform | Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.000021 | - |
- |
Homo sapiens | rolipram | |
0.000042 | - |
- |
Homo sapiens | Ro20-1724 | |
0.0059 | - |
- |
Homo sapiens | 3-isobuytl-1-methylxanthine |