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Literature summary for 3.1.4.52 extracted from

  • Zheng, Y.; Tsuji, G.; Opoku-Temeng, C.; Sintim, H.O.
    Inhibition of P. aeruginosa c-di-GMP phosphodiesterase RocR and swarming motility by a benzoisothiazolinone derivative (2016), Chem. Sci., 7, 6238-6244 .
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
N-(4-hydroxyphenyl)-4-(3-oxo-1,2-benzothiazol-2(3H)-yl)butanamide compound inhibits Pseudomonas. aeruginosa (PAO1) swarming but not swimming or biofilm formation, it does not inhibit other Pseudomonas aeruginosa phosphodiesterases, such as DipA, PvrR and PA4108 Pseudomonas aeruginosa

Organism

Organism UniProt Comment Textmining
Pseudomonas aeruginosa Q9HX69
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Pseudomonas aeruginosa ATCC 15692 Q9HX69
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Synonyms

Synonyms Comment Organism
PA3947
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Pseudomonas aeruginosa
RocR
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Pseudomonas aeruginosa