Activating Compound | Comment | Organism | Structure |
---|---|---|---|
phosphatidylinositol 3,4,5-trisphosphate | increases PLD activity | Homo sapiens | |
phosphatidylinositol 4,5-bisphosphate | activates | Homo sapiens | |
phosphatidylinositol-3,4,5-trisphosphate | with partially purified enzyme, stimulation up to 5fold | Homo sapiens | |
phosphatidylinositol-4,5-bisphosphate | in native myocardium, stimulation up to 2fold at 0.1 mM, accompanied by increase in diacylglycerol, with partially purified enzyme, stimulation up to 10fold at 0.1 mM | Homo sapiens |
Cloned (Comment) | Organism |
---|---|
- |
Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
neomycin | inhibitory in native myocardium, where phosphatidylinositol-4,5-bisphosphate restores, not inhibitory with partially purified enzyme; inhibits activity in human atrial myocardium, but has no effect on the activity of partially solubilized enzyme | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Homo sapiens | Q13393 | isozyme PLD1 | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
heart | atrial myocardium | Homo sapiens | - |
myocardium | - |
Homo sapiens | - |