Inhibitors | Comment | Organism | Structure |
---|---|---|---|
4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone | Ro20-1724 | Cavia porcellus | |
cGMP | - |
Cavia porcellus | |
Milrinone | - |
Cavia porcellus | |
quercetin | - |
Cavia porcellus | |
quercetin-3,5,7,3',4'-O-pentaacetate | - |
Cavia porcellus | |
quercetin-3,5,7,3',4'-O-pentamethylether | - |
Cavia porcellus | |
quercetin-3,7,3',4'-O-tetramethylether | - |
Cavia porcellus | |
quercetin-3,7,4'-O-trimethylether | ayanin | Cavia porcellus | |
quercetin-3-O-methyl-5,7,3',4'-O-tetraacetate | - |
Cavia porcellus | |
quercetin-3-O-methylether | - |
Cavia porcellus | |
rolipram | - |
Cavia porcellus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Cavia porcellus | - |
- |
- |
Purification (Comment) | Organism |
---|---|
partially purified by Q-Sepharose column chromatography | Cavia porcellus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
heart | - |
Cavia porcellus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
nucleoside 3',5'-cyclic phosphate + H2O | - |
Cavia porcellus | nucleoside 5'-phosphate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PDE3 | - |
Cavia porcellus |
phosphodiesterase-3 | - |
Cavia porcellus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0008 | - |
PDE3 | Cavia porcellus | quercetin-3-O-methyl-5,7,3',4'-O-tetraacetate | |
0.0016 | - |
PDE3 | Cavia porcellus | quercetin-3-O-methylether | |
0.002 | - |
PDE3 | Cavia porcellus | Milrinone | |
0.002 | - |
PDE3 | Cavia porcellus | quercetin-3,5,7,3',4'-O-pentaacetate | |
0.0041 | - |
PDE3 | Cavia porcellus | quercetin-3,7,4'-O-trimethylether | |
0.0047 | - |
PDE3 | Cavia porcellus | quercetin-3,5,7,3',4'-O-pentamethylether | |
0.0056 | - |
PDE3 | Cavia porcellus | quercetin | |
0.0228 | - |
PDE3 | Cavia porcellus | quercetin-3,7,3',4'-O-tetramethylether | |
0.0869 | - |
PDE3 | Cavia porcellus | quercetin-3-O-methylether |