Inhibitors | Comment | Organism | Structure |
---|---|---|---|
3',5'-cAMP | IC50: above 0.5 mM | Homo sapiens | |
5-adenoylimino phosphate | IC50: above 0.5 mM | Homo sapiens | |
adeno 5'-diphosphate | IC50: above 0.5 mM | Homo sapiens | |
adeno-2',3'-cyclic phospho 5'-monophosphate | IC50: 0.2 mM | Homo sapiens | |
adeno-2',3'-cyclic phospho 5'-phosphosulfate | IC50: 0.5 mM | Homo sapiens | |
ADP | IC50: 0.3 mM | Homo sapiens | |
AMP | IC50: 0.08 mM, non-competitive inhibition | Homo sapiens | |
ATP | IC50: 0.8 mM | Homo sapiens | |
lysophosphatidic acid | IC50: 0.04 mM | Homo sapiens | |
NAD+ | IC50: above 0.5 mM | Homo sapiens | |
NADP+ | IC50: above 0.5 mM | Homo sapiens | |
phosphate | IC50: 10 mM, non-competitive inhibition | Homo sapiens | |
phosphatidyl-myo-inositol 3,4,5-triphosphate | IC50: 0.003 mM | Homo sapiens | |
phosphatidyl-myo-inositol 4,5-diphosphate | IC50: 0.25 mM | Homo sapiens | |
phosphatidylcholine | IC50: 2 mM | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
HOG cell | human oligodendroglioma cell | Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
6-hexadecanoylamino-4-methylumbelliferyl-phosphocholine + H2O | - |
Homo sapiens | 6-hexadecanoylamino-4-methylumbelliferone + choline phosphate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
aSMase | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.003 | - |
IC50: 0.003 mM | Homo sapiens | phosphatidyl-myo-inositol 3,4,5-triphosphate | |
0.04 | - |
IC50: 0.04 mM | Homo sapiens | lysophosphatidic acid | |
0.08 | - |
IC50: 0.08 mM, non-competitive inhibition | Homo sapiens | AMP | |
0.2 | - |
IC50: 0.2 mM | Homo sapiens | adeno-2',3'-cyclic phospho 5'-monophosphate | |
0.25 | - |
IC50: 0.25 mM | Homo sapiens | phosphatidyl-myo-inositol 4,5-diphosphate | |
0.3 | - |
IC50: 0.3 mM | Homo sapiens | ADP | |
0.5 | - |
IC50: 0.5 mM | Homo sapiens | adeno-2',3'-cyclic phospho 5'-phosphosulfate | |
0.5 | - |
IC50: above 0.5 mM | Homo sapiens | NAD+ | |
0.5 | - |
IC50: above 0.5 mM | Homo sapiens | NADP+ | |
0.5 | - |
IC50: above 0.5 mM | Homo sapiens | 3',5'-cAMP | |
0.5 | - |
IC50: above 0.5 mM | Homo sapiens | adeno 5'-diphosphate | |
0.5 | - |
IC50: above 0.5 mM | Homo sapiens | 5-adenoylimino phosphate | |
0.8 | - |
IC50: 0.8 mM | Homo sapiens | ATP | |
2 | - |
IC50: 2 mM | Homo sapiens | phosphatidylcholine | |
10 | - |
IC50: 10 mM, non-competitive inhibition | Homo sapiens | phosphate |