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Literature summary for 3.1.3.2 extracted from

  • Mohd-Pahmi, S.H.; Hussein, W.M.; Schenk, G.; McGeary, R.P.
    Synthesis, modelling and kinetic assays of potent inhibitors of purple acid phosphatase (2011), Bioorg. Med. Chem. Lett., 21, 3092-3094.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
[(butanoylamino)(naphthalen-1-yl)methyl]phosphonic acid
-
Phaseolus vulgaris
[(butanoylamino)(naphthalen-1-yl)methyl]phosphonic acid
-
Sus scrofa
[(decanoylamino)(naphthalen-1-yl)methyl]phosphonic acid
-
Phaseolus vulgaris
[(decanoylamino)(naphthalen-1-yl)methyl]phosphonic acid
-
Sus scrofa
[(dodecanoylamino)(naphthalen-1-yl)methyl]phosphonic acid
-
Phaseolus vulgaris
[(dodecanoylamino)(naphthalen-1-yl)methyl]phosphonic acid
-
Sus scrofa
[(heptanoylamino)(naphthalen-1-yl)methyl]phosphonic acid
-
Phaseolus vulgaris
[(heptanoylamino)(naphthalen-1-yl)methyl]phosphonic acid
-
Sus scrofa
[(hexadecanoylamino)(naphthalen-1-yl)methyl]phosphonic acid
-
Phaseolus vulgaris
[(hexadecanoylamino)(naphthalen-1-yl)methyl]phosphonic acid
-
Sus scrofa
[naphthalen-1-yl(octanoylamino)methyl]phosphonic acid
-
Phaseolus vulgaris
[naphthalen-1-yl(octanoylamino)methyl]phosphonic acid
-
Sus scrofa
[naphthalen-1-yl(tetradecanoylamino)methyl]phosphonic acid
-
Phaseolus vulgaris
[naphthalen-1-yl(tetradecanoylamino)methyl]phosphonic acid
-
Sus scrofa

Organism

Organism UniProt Comment Textmining
Phaseolus vulgaris
-
-
-
Sus scrofa
-
-
-

Synonyms

Synonyms Comment Organism
acid phosphatase
-
Sus scrofa
PAP
-
Sus scrofa
rkbPAP red kidney bean PAP Phaseolus vulgaris

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.005
-
[(dodecanoylamino)(naphthalen-1-yl)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Phaseolus vulgaris
0.008
-
[naphthalen-1-yl(tetradecanoylamino)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Sus scrofa
0.01
-
[(decanoylamino)(naphthalen-1-yl)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Sus scrofa
0.011
-
[naphthalen-1-yl(tetradecanoylamino)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Phaseolus vulgaris
0.013
-
[(hexadecanoylamino)(naphthalen-1-yl)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Sus scrofa
0.021
-
[(dodecanoylamino)(naphthalen-1-yl)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Sus scrofa
0.031
-
[(hexadecanoylamino)(naphthalen-1-yl)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Phaseolus vulgaris
0.044
-
[naphthalen-1-yl(octanoylamino)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Sus scrofa
0.057
-
[(decanoylamino)(naphthalen-1-yl)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Phaseolus vulgaris
0.116
-
[(heptanoylamino)(naphthalen-1-yl)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Sus scrofa
0.195
-
[naphthalen-1-yl(octanoylamino)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Phaseolus vulgaris
0.222
-
[(heptanoylamino)(naphthalen-1-yl)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Phaseolus vulgaris
0.238
-
[(butanoylamino)(naphthalen-1-yl)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Phaseolus vulgaris
0.363
-
[(butanoylamino)(naphthalen-1-yl)methyl]phosphonic acid pH 4.9, competitive inhibition constant, temperature not specified in the publication Sus scrofa