Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(2Z)-2-(benzoylamino)-3-[2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]prop-2-enoate | with 0.1 mM 35% remaining activity | Bos taurus | |
(4-methoxyphenyl)[2-(4-methoxyphenyl)-1-benzothiophen-3-yl]methanone | with 0.1 mM 70% remaining activity | Bos taurus | |
1-(2-phenyl-1-benzothiophen-3-yl)methanamine | with 0.4 mM 76% remaining activity | Sus scrofa | |
1-benzothiophen-3-yl 4-fluorophenyl ether | with 0.4 mM 78% remaining activity | Sus scrofa | |
1-benzothiophen-3-yl(4-methoxyphenyl)methanone | with 0.1 mM 40% remaining activity | Bos taurus | |
1-benzothiophen-3-yl(phenyl)methanone | with 0.1 mM 43% remaining activity | Bos taurus | |
2-(1-benzothiophen-2-yl)aniline | with 0.4 mM 70% remaining activity | Sus scrofa | |
2-(2-chlorophenyl)-1-benzothiophene-3-carbaldehyde | with 0.1 mM 63% remaining activity | Bos taurus | |
2-(2-methylphenyl)-1-benzothiophene-3-carbonitrile | with 0.1 mM 5% remaining activity | Bos taurus | |
2-(2-nitrophenyl)-1-benzothiophene-3-carbaldehyde | with 0.4 mM 78% remaining activity | Sus scrofa | |
2-(3-chlorophenyl)-1-benzothiophene-3-carbaldehyde | with 0.1 mM 62% remaining activity | Bos taurus | |
2-(3-formyl-1-benzothiophen-2-yl)benzonitrile | with 0.4 mM 79% remaining activity | Sus scrofa | |
2-(3-methoxy-1-benzothiophen-2-yl)benzonitrile | with 0.1 mM 57% remaining activity | Bos taurus | |
2-(3-methoxy-1-benzothiophen-2-yl)benzonitrile | with 0.4 mM 79% remaining activity | Sus scrofa | |
2-(3-pyridine)-3-oxime-benzo[b]thiophene | with 0.4 mM 71% remaining activity | Sus scrofa | |
2-(4-chlorophenyl)-1-benzothiophene-3-carbaldehyde | with 0.1 mM 9% remaining activity | Bos taurus | |
2-(4-chlorophenyl)-1-benzothiophene-3-carbonitrile | with 0.1 mM 69% remaining activity | Bos taurus | |
2-(4-methoxyphenyl)-1-benzothiophene-3-carbaldehyde | with 0.1 mM 37% remaining activity | Bos taurus | |
2-(naphthalen-2-yl)-1-benzothiophene-3-carbonitrile | with 0.1 mM 18% remaining activity | Bos taurus | |
2-(pyridin-3-yl)-1-benzothiophene-3-carbaldehyde | with 0.4 mM 79% remaining activity | Sus scrofa | |
2-iodo-1-benzothiophene | with 0.1 mM 41% remaining activity | Bos taurus | |
2-iodo-1-benzothiophene | with 0.4 mM 54% remaining activity | Sus scrofa | |
2-phenyl-1-benzothiophene-3-carbaldehyde | with 0.1 mM 41% remaining activity | Bos taurus | |
2-phenyl-1-benzothiophene-3-carbaldehyde | with 0.4 mM 77% remaining activity | Sus scrofa | |
2-phenyl-1-benzothiophene-3-carbonitrile | with 0.1 mM 76% remaining activity | Bos taurus | |
2-phenyl-3-oxime-benzo[b]thiophene | with 0.1 mM 1% remaining activity | Bos taurus | |
2-phenyl-3-oxime-benzo[b]thiophene | with 0.4 mM 68% remaining activity | Sus scrofa | |
2-phenyl-benzo[b]thiophene-3-carboxylic acid | with 0.4 mM 78% remaining activity | Sus scrofa | |
2-[3-(2,2,2-trifluoroethyl)-1-benzothiophen-2-yl]benzonitrile | with 0.1 mM 70% remaining activity | Bos taurus | |
2-[3-(4-chlorophenoxy)-1-benzothiophen-2-yl]benzonitrile | with 0.4 mM 79% remaining activity | Sus scrofa | |
2-[3-(4-fluorophenoxy)-1-benzothiophen-2-yl]benzonitrile | with 0.1 mM 66% remaining activity | Bos taurus | |
2-[4-(1-benzothiophen-3-yl)piperazin-1-yl]phenol | with 0.1 mM 49% remaining activity | Bos taurus | |
2-[4-(trifluoromethyl)phenyl]-1-benzothiophene-3-carbaldehyde | with 0.1 mM 30% remaining activity | Bos taurus | |
3-(3-methoxy-1-benzothiophen-2-yl)pyridine | with 0.4 mM 44% remaining activity | Sus scrofa | |
3-(3-methoxy-1-benzothiophen-2-yl)quinoline | with 0.1 mM 64% remaining activity | Bos taurus | |
3-(4-fluorophenoxy)-1-benzothiophene 1-oxide | with 0.4 mM 79% remaining activity | Sus scrofa | |
3-methoxy-2-(2-methylphenyl)-1-benzothiophene | with 0.1 mM 73% remaining activity | Bos taurus | |
3-methoxy-2-(4-methoxyphenyl)-1-benzothiophene | with 0.1 mM 78% remaining activity | Bos taurus | |
4-(1-benzothiophen-3-yloxy)benzaldehyde | with 0.1 mM 9% remaining activity | Bos taurus | |
4-[(1-oxido-1-benzothiophen-3-yl)oxy]benzonitrile | with 0.4 mM 67% remaining activity | Sus scrofa | |
6-(1-benzothiophen-3-yl)-2,3,5,6-tetrahydroimidazo[2,1-b][1,3]thiazole | with 0.4 mM 19% remaining activity | Sus scrofa | |
6-(1-benzothiophen-3-yl)-5,6-dihydroimidazo[2,1-b][1,3]thiazole | with 0.4 mM 11% remaining activity | Sus scrofa | |
levamisole | with 0.4 mM 10% remaining activity | Sus scrofa | |
methyl (2E)-2-(benzoylamino)-3-[2-(4-methoxyphenyl)-1-benzothiophen-3-yl]prop-2-enoate | with 0.1 mM 77% remaining activity | Bos taurus | |
methyl 3-(1-benzothiophen-3-yl)-N-benzoylalaninate | with 0.4 mM 74% remaining activity | Sus scrofa | |
methyl N-benzoyl-3-[2-[4-(trifluoromethyl)phenyl]-1-benzothiophen-3-yl]alaninate | with 0.1 mM 63% remaining activity | Bos taurus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
- |
- |
Sus scrofa | - |
domestica | - |
Purification (Comment) | Organism |
---|---|
commercial product | Sus scrofa |
commercial product | Bos taurus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
intestine | - |
Bos taurus | - |
kidney | - |
Sus scrofa | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
4-nitrophenyl phosphate + H2O | - |
Sus scrofa | 4-nitrophenol + phosphate | - |
? | |
4-nitrophenyl phosphate + H2O | - |
Bos taurus | 4-nitrophenol + phosphate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
alkaline phosphatase | - |
Sus scrofa |
alkaline phosphatase | - |
Bos taurus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.085 | - |
6-(1-benzothiophen-3-yl)-5,6-dihydroimidazo[2,1-b][1,3]thiazole | - |
Sus scrofa | |
0.093 | - |
levamisole | - |
Sus scrofa | |
0.135 | - |
6-(1-benzothiophen-3-yl)-2,3,5,6-tetrahydroimidazo[2,1-b][1,3]thiazole | - |
Sus scrofa |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
additional information | - |
aus tab | Sus scrofa | additional information |