Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 3.1.1.8 extracted from

  • Graham, S.G.; Crossley, A.W.A.
    The characteristics of the inhibition of serum cholinesterase by metoclopramide (1995), Eur. J. Clin. Pharmacol., 48, 225-228.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
metoclopramide 0.001-0.0019 mM, 50% competitive inhibition Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
serum
-
Homo sapiens
-

Synonyms

Synonyms Comment Organism
choline esterase
-
Homo sapiens

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.001 0.0019 metoclopramide competitive inhibition Homo sapiens