Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 3.1.1.7 extracted from

  • Cibickova, L.; Radomir, H.; Stanislav, M.; Norbert, C.; Helena, Z.; Daniel, J.; Alena, T.; Eva, B.; Vladimir, P.
    The influence of simvastatin, atorvastatin and high-cholesterol diet on acetylcholinesterase activity, amyloid beta and cholesterol synthesis in rat brain (2009), Steroids, 74, 13-19.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
additional information acetylcholinesterase activity remains unaffected by the two drugs simvastatin and atorvastatin, that reduce brain lathosterol and cholesterol synthesis rate but do not reduce cholesterol levels, overview Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
additional information acetylcholinesterase activity remains unaffected by the two drugs simvastatin and atorvastatin, that reduce brain lathosterol and cholesterol synthesis rate but do not reduce cholesterol levels, overview Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
male Wistar rats
-

Source Tissue

Source Tissue Comment Organism Textmining
brain
-
Rattus norvegicus
-

Specific Activity [micromol/min/mg]

Specific Activity Minimum [µmol/min/mg] Specific Activity Maximum [µmol/min/mg] Comment Organism
additional information
-
-
Rattus norvegicus

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
S-acetylthiocholine + H2O detection with 5,5'-dithio-bis-2-nitrobenzoic acid, i.e. DTNB Rattus norvegicus acetate + thiocholine
-
?

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
25
-
assay at Rattus norvegicus

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.6
-
assay at Rattus norvegicus