Inhibitors | Comment | Organism | Structure |
---|---|---|---|
3-(2-bromoethoxy)-4-chloro-7-nitro-1H-isochromen-1-one | - |
Sus scrofa | |
3-(2-bromoethoxy)-7-nitro-1H-isochromen-1-one | - |
Sus scrofa | |
3-(2-cyclohexylethoxy)-4-trifluoroacetylisocoumarin | - |
Sus scrofa | |
3-(2-cyclohexylethoxy)-7-nitroisocoumarin | - |
Sus scrofa | |
3-(3-bromopropoxy)-4-chloro-7-nitro-1H-isochromen-1-one | - |
Sus scrofa | |
3-(3-bromopropoxy)-7-nitro-1H-isochromen-1-one | - |
Sus scrofa | |
3-butoxy-4-chloroisocoumarin | - |
Sus scrofa | |
3-cyclohexylmethoxy-7-nitroisocoumarin | - |
Sus scrofa | |
3-cyclohexylmethyl-4-(trifluoroacetyl)isocoumarin | - |
Sus scrofa | |
3-propoxy-4-(trifluoroacetyl)isocoumarin | - |
Sus scrofa | |
4-chloro-3-(2-cyclohexylethoxy)-7-nitroisocoumarin | - |
Sus scrofa | |
4-chloro-3-(2-cyclohexylethoxy)isocoumarin | - |
Sus scrofa | |
4-chloro-3-(2-cyclopentylethoxy)isocoumarin | - |
Sus scrofa | |
4-chloro-3-(3-cyclohexylpropoxy)isocoumarin | - |
Sus scrofa | |
4-chloro-3-(3-cyclopentylpropoxy)isocoumarin | potent reversible inhibitor | Sus scrofa | |
4-chloro-3-(4-cyclohexylbutoxy)isocoumarin | potent reversible inhibitor | Sus scrofa | |
4-chloro-3-(4-cyclohexylcyclohexyloxy)isocoumarin | - |
Sus scrofa | |
4-chloro-3-(5-cyclohexylpentoxy)isocoumarin | - |
Sus scrofa | |
4-chloro-3-(cyclohexylmethoxy)isocoumarin | - |
Sus scrofa | |
4-chloro-3-(cyclopentylmethoxy)isocoumarin | - |
Sus scrofa | |
4-chloro-3-(cyclopentyloxy)isocoumarin | - |
Sus scrofa | |
4-chloro-3-cyclohexylmethoxy-7-nitroisocoumarin | - |
Sus scrofa | |
4-chloro-3-methoxy-7-nitroisocoumarin | - |
Sus scrofa | |
4-chloro-3-propoxyisocoumarin | - |
Sus scrofa | |
4-chloro-7-cyclohexanecarboxamide-3-methoxyisocoumarin | - |
Sus scrofa | |
7-amino-3-(2-bromoethoxy)-4-chloro-1H-isochromen-1-one | - |
Sus scrofa | |
7-amino-3-(2-bromoethoxy)isocoumarin | - |
Sus scrofa | |
7-amino-4-chloro-3-methoxyisocoumarin | - |
Sus scrofa | |
7-benzamido-4-chloro-3-methoxyisocoumarin | - |
Sus scrofa |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Sus scrofa | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
pancreas | - |
Sus scrofa | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
cholesteryl linoleate + H2O | - |
Sus scrofa | cholesterol + linoleate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
bile salt-dependent lipase | - |
Sus scrofa |
bile salt-stimulated lipase | - |
Sus scrofa |
Carboxyl ester lipase | - |
Sus scrofa |
CEase | - |
Sus scrofa |
nonspecific lipase | - |
Sus scrofa |
pancreatic cholesterol esterase | - |
Sus scrofa |
Pancreatic lysophospholipase | - |
Sus scrofa |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000011 | - |
4-chloro-3-(4-cyclohexylbutoxy)isocoumarin | - |
Sus scrofa | |
0.000019 | - |
4-chloro-3-(3-cyclopentylpropoxy)isocoumarin | - |
Sus scrofa | |
0.00018 | - |
4-chloro-3-(3-cyclohexylpropoxy)isocoumarin | - |
Sus scrofa | |
0.00019 | - |
4-chloro-3-(4-cyclohexylcyclohexyloxy)isocoumarin | - |
Sus scrofa | |
0.00026 | - |
4-chloro-3-(2-cyclopentylethoxy)isocoumarin | - |
Sus scrofa | |
0.00036 | - |
4-chloro-3-(cyclopentylmethoxy)isocoumarin | - |
Sus scrofa | |
0.0007 | - |
4-chloro-3-(2-cyclohexylethoxy)-7-nitroisocoumarin | - |
Sus scrofa | |
0.00095 | - |
4-chloro-3-(cyclopentyloxy)isocoumarin | - |
Sus scrofa | |
0.0012 | - |
4-chloro-3-(4-cyclohexylbutoxy)isocoumarin | - |
Sus scrofa | |
0.0012 | - |
4-chloro-3-(2-cyclohexylethoxy)isocoumarin | - |
Sus scrofa | |
0.0018 | - |
4-chloro-3-(cyclohexylmethoxy)isocoumarin | - |
Sus scrofa | |
0.0036 | - |
4-chloro-3-propoxyisocoumarin | - |
Sus scrofa | |
0.0057 | - |
4-chloro-3-cyclohexylmethoxy-7-nitroisocoumarin | - |
Sus scrofa | |
0.0065 | - |
3-butoxy-4-chloroisocoumarin | - |
Sus scrofa | |
0.017 | - |
7-amino-4-chloro-3-methoxyisocoumarin | - |
Sus scrofa | |
0.019 | - |
4-chloro-3-methoxy-7-nitroisocoumarin | - |
Sus scrofa | |
0.025 | - |
3-propoxy-4-(trifluoroacetyl)isocoumarin | Ki above 0.025 mM | Sus scrofa | |
0.025 | - |
4-chloro-7-cyclohexanecarboxamide-3-methoxyisocoumarin | Ki above 0.025 mM | Sus scrofa | |
0.054 | - |
3-cyclohexylmethoxy-7-nitroisocoumarin | - |
Sus scrofa | |
0.062 | - |
4-chloro-3-(5-cyclohexylpentoxy)isocoumarin | - |
Sus scrofa | |
0.073 | - |
3-(2-cyclohexylethoxy)-4-trifluoroacetylisocoumarin | - |
Sus scrofa | |
0.1 | - |
3-cyclohexylmethyl-4-(trifluoroacetyl)isocoumarin | Ki above 0.1 mM | Sus scrofa | |
0.1 | - |
3-(2-cyclohexylethoxy)-7-nitroisocoumarin | Ki above 0.1 mM | Sus scrofa | |
0.1 | - |
7-amino-3-(2-bromoethoxy)isocoumarin | Ki above 0.1 mM | Sus scrofa | |
0.25 | - |
7-benzamido-4-chloro-3-methoxyisocoumarin | Ki above 0.25 mM | Sus scrofa |