Activating Compound | Comment | Organism | Structure |
---|---|---|---|
additional information | no activation by adenine nucleotides | Rattus norvegicus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Cd2+ | 5 mM, strong inhibition | Rattus norvegicus | |
dehydroepiandrosterone | cortisol as substrate; kinetics | Rattus norvegicus | |
dexamethasone | cortisol as substrate; kinetics | Rattus norvegicus | |
diethylstilbestrol | cortisol as substrate | Rattus norvegicus | |
additional information | no inhibition by adenine nucleotides | Rattus norvegicus | |
progesterone | cortisol as substrate | Rattus norvegicus | |
Zn2+ | 5 mM, strong inhibition | Rattus norvegicus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00628 | - |
3'-phosphoadenylylsulfate | pH 6.8, 37.5°C | Rattus norvegicus | |
0.00682 | - |
cortisol | pH 6.8, 37.5°C | Rattus norvegicus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
cytosol | - |
Rattus norvegicus | 5829 | - |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Ba2+ | activation | Rattus norvegicus | |
Ba2+ | 5 mM | Rattus norvegicus | |
Ba2+ | in decreasing order of efficiency: Mn2+, Cr2+, Co2+, Mg2+, Ba2+, Ca2+, Ni2+ | Rattus norvegicus | |
Ca2+ | activation | Rattus norvegicus | |
Ca2+ | 5 mM | Rattus norvegicus | |
Ca2+ | in decreasing order of efficiency: Mn2+, Cr2+, Co2+, Mg2+, Ba2+, Ca2+, Ni2+ | Rattus norvegicus | |
Co2+ | activation | Rattus norvegicus | |
Co2+ | 5 mM | Rattus norvegicus | |
Co2+ | in decreasing order of efficiency: Mn2+, Cr2+, Co2+, Mg2+, Ba2+, Ca2+, Ni2+ | Rattus norvegicus | |
Cr2+ | activation | Rattus norvegicus | |
Cr2+ | 5 mM | Rattus norvegicus | |
Cr2+ | in decreasing order of efficiency: Mn2+, Cr2+, Co2+, Mg2+, Ba2+, Ca2+, Ni2+ | Rattus norvegicus | |
Mg2+ | activation | Rattus norvegicus | |
Mg2+ | 5 mM | Rattus norvegicus | |
Mg2+ | in decreasing order of efficiency: Mn2+, Cr2+, Co2+, Mg2+, Ba2+, Ca2+, Ni2+ | Rattus norvegicus | |
Mn2+ | activation | Rattus norvegicus | |
Mn2+ | 5 mM | Rattus norvegicus | |
Mn2+ | in decreasing order of efficiency: Mn2+, Cr2+, Co2+, Mg2+, Ba2+, Ca2+, Ni2+ | Rattus norvegicus | |
Ni2+ | activation | Rattus norvegicus | |
Ni2+ | 5 mM | Rattus norvegicus | |
Ni2+ | in decreasing order of efficiency: Mn2+, Cr2+, Co2+, Mg2+, Ba2+, Ca2+, Ni2+ | Rattus norvegicus |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
61500 | - |
sulfotransferase III, gel filtration | Rattus norvegicus |
65000 | - |
sedimentation velocity experiments | Rattus norvegicus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
3'-phosphoadenylylsulfate + cortisol | Rattus norvegicus | - |
adenosine 3',5'-bisphosphate + cortisol 21-sulfate | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | - |
male CDR Fisher rats | - |
Purification (Comment) | Organism |
---|---|
partial | Rattus norvegicus |
sulfotransferase III | Rattus norvegicus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
blood | - |
Rattus norvegicus | - |
liver | - |
Rattus norvegicus | - |
additional information | tissue distribution | Rattus norvegicus | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
0.00098 | - |
- |
Rattus norvegicus |
Storage Stability | Organism |
---|---|
-20°C, at least 3 months | Rattus norvegicus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
3'-phosphoadenylylsulfate + cortisol | - |
Rattus norvegicus | adenosine 3',5'-bisphosphate + cortisol 21-sulfate | - |
? | |
3'-phosphoadenylylsulfate + cortisol | i.e. PAPS, glucocorticoids are preferred substrates | Rattus norvegicus | adenosine 3',5'-bisphosphate + cortisol 21-sulfate | - |
? | |
3'-phosphoadenylylsulfate + dehydroepiandrosterone | - |
Rattus norvegicus | adenosine 3',5'-bisphosphate + ? | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37.5 | - |
assay at | Rattus norvegicus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
6 | - |
cortisol as substrate | Rattus norvegicus |