Inhibitors | Comment | Organism | Structure |
---|---|---|---|
adenosine 3',5'-bisphosphate | - |
Homo sapiens | |
ATP | M-PST | Homo sapiens | |
NaCl | 50% inhibition at: 325 mM; M-PST | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00035 | - |
3'-phosphoadenylylsulfate | M-PST, pH 7.0, 37°C | Homo sapiens | |
0.0029 | - |
dopamine | M-PST, pH 7.0, 37°C | Homo sapiens |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
250000 | - |
isozyme M-PST, gel filtration | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
2 forms: simple phenol sulfating P-PST, monoamine sulfating M-PST | - |
Purification (Comment) | Organism |
---|---|
monoamine-sulfating form, M-PST | Homo sapiens |
Reaction | Comment | Organism | Reaction ID |
---|---|---|---|
3'-phosphoadenylyl sulfate + a phenol = adenosine 3',5'-bisphosphate + an aryl sulfate | isozyme M-PST: ordered bisubstrate reaction mechanism | Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
brain | - |
Homo sapiens | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
- |
Homo sapiens |
0.0077 | - |
purified M-PST | Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
3'-phosphoadenylyl sulfate + a phenol | - |
Homo sapiens | adenosine 3',5'-bisphosphate + an aryl sulfate | - |
? | |
3'-phosphoadenylylsulfate + 4-methoxytyramine | - |
Homo sapiens | adenosine 3',5'-bisphosphate + ? | - |
? | |
3'-phosphoadenylylsulfate + dopamine | - |
Homo sapiens | adenosine 3',5'-bisphosphate + ? | - |
? | |
3'-phosphoadenylylsulfate + tyramine | - |
Homo sapiens | adenosine 3',5'-bisphosphate + tyramine O-sulfate | - |
? | |
additional information | substrate specificity | Homo sapiens | ? | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7 | - |
M-PST, with substrate dopamine | Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00007 | - |
adenosine 3',5'-bisphosphate | M-PST, pH 7.0, 37°C | Homo sapiens | |
0.18 | - |
ATP | M-PST, pH 7.0, 37°C | Homo sapiens |