Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 2.7.7.31 extracted from

  • Di Santo, R.; Maga, G.
    Human terminal deoxynucleotidyl transferases as novel targets for anticancer chemotherapy (2006), Curr. Med. Chem., 13, 2353-2368.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
(1R,2S)-1-(6-aminopurin-9-yl)-2-(Hydroxymethyl)cyclopentane
-
Homo sapiens
3'-azido-TTP
-
Homo sapiens
Ap5A
-
Homo sapiens
cordycepin selectively cytotoxic against TdT+ leukemic cells, particularly in combination with the adenosine deaminase inhibitor deoxycoformycin Homo sapiens
D-/L-carbocyclic dideoxynucleoside triphosphates
-
Homo sapiens
ddATP
-
Homo sapiens
ddCTP
-
Homo sapiens
ddGTP
-
Homo sapiens
ddTTP
-
Homo sapiens
P1,P5-diadenosine 5'-pentaphosphate
-
Homo sapiens

Metals/Ions

Metals/Ions Comment Organism Structure
Co2+
-
Mus musculus
Co2+
-
Homo sapiens
Mg2+
-
Mus musculus
Mg2+
-
Homo sapiens
Mn2+
-
Mus musculus
Mn2+
-
Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
bone marrow
-
Homo sapiens
-
thymus
-
Homo sapiens
-

Synonyms

Synonyms Comment Organism
terminal deoxynucleotidyl transferase
-
Homo sapiens
terminal deoxynucleotidyl transferase (TDT)
-
Mus musculus

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.00025
-
Ap5A
-
Homo sapiens
0.0005
-
(1R,2S)-1-(6-aminopurin-9-yl)-2-(Hydroxymethyl)cyclopentane
-
Homo sapiens
0.0009 0.006 cordycepin
-
Homo sapiens
0.0013
-
ddATP
-
Homo sapiens
0.0013
-
ddGTP
-
Homo sapiens
0.0028
-
ddCTP
-
Homo sapiens
0.005 0.01 D-/L-carbocyclic dideoxynucleoside triphosphates
-
Homo sapiens
0.01
-
3'-azido-TTP
-
Homo sapiens
0.0175
-
ddTTP
-
Homo sapiens