Inhibitors | Comment | Organism | Structure |
---|---|---|---|
5'-fluorosulfonylbenzoyladenosine | - |
Brassica oleracea | |
mammalian protein phosphatase 2C | - |
Brassica oleracea |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.013 | - |
HMRSAMSGLHGVKRR | pH 7.0, 30°C, kinase A | Brassica oleracea | |
0.034 | - |
HMRSAMTGLHGVKRR | pH 7.0, 30°C, kinase A | Brassica oleracea | |
0.038 | - |
HMRSAMSGLHLGKRR | pH 7.0, 30°C, kinase A | Brassica oleracea | |
0.0404 | - |
HGRSAMSGLHLVKRR | pH 7.0, 30°C, kinase A | Brassica oleracea | |
0.042 | - |
HMRSAMSGLHLGKRR | pH 7.0, 30°C, kinase B | Brassica oleracea | |
0.049 | - |
HMRSAMSGLHGGKRR | pH 7.0, 30°C, kinase A | Brassica oleracea | |
0.0498 | - |
HMRSAMSGLHLVKRR | pH 7.0, 30°C, kinase A | Brassica oleracea | |
0.065 | - |
HMRSAMTGLHGVKRR | pH 7.0, 30°C, kinase B | Brassica oleracea | |
0.069 | - |
HMRSAGSGLHLVKRR | pH 7.0, 30°C, kinase B | Brassica oleracea | |
0.07 | - |
HMRSAGSGLHLVKRR | pH 7.0, 30°C, kinase A | Brassica oleracea | |
0.091 | - |
HMRSAMSGLHLVKRR | pH 7.0, 30°C, kinase B | Brassica oleracea | |
0.096 | - |
HMRSAMSGLHGVKRR | pH 7.0, 30°C, kinase B | Brassica oleracea | |
0.111 | - |
HMKSAMSGLHLVKRR | pH 7.0, 30°C, kinase B | Brassica oleracea | |
0.118 | - |
HMHSAMSGLHLVKRR | pH 7.0, 30°C, kinase A | Brassica oleracea | |
0.133 | - |
HMKSAMSGLHLVKRR | pH 7.0, 30°C, kinase A | Brassica oleracea | |
0.428 | - |
HMHSAMSGLHLVKRR | pH 7.0, 30°C, kinase B | Brassica oleracea | |
0.573 | - |
HMGSAMSGLHLVKRR | pH 7.0, 30°C, kinase A | Brassica oleracea | |
2.316 | - |
HMGSAMSGLHLVKRR | pH 7.0, 30°C, kinase B | Brassica oleracea |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
45000 | - |
major form B, gel filtration | Brassica oleracea |
58000 | - |
x * 58000, catalytic subunit | Brassica oleracea |
150000 | - |
major form A, electrophoresis in non-denaturing gels | Brassica oleracea |
160000 | - |
major form A, PAGE | Brassica oleracea |
200000 | - |
major form A, gel filtration | Brassica oleracea |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + [hydroxymethylglutaryl-CoA reductase (NADPH)] | Brassica oleracea | inactivates EC 1.1.1.34 by phosphorylation | ADP + [hydroxymethylglutaryl-CoA reductase (NADPH)] phosphate | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Brassica oleracea | - |
cauliflower, var. botrytis | - |
Purification (Comment) | Organism |
---|---|
2 isoformes, major form A and major form B | Brassica oleracea |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
inflorescence | - |
Brassica oleracea | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
3.281 | - |
major form B | Brassica oleracea |
13.1 | - |
major form A | Brassica oleracea |
Storage Stability | Organism |
---|---|
-70°C, 0.5 mg protein/ml, frozen in liquid nitrogen, can be stored with no loss of activity | Brassica oleracea |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + HGRSAMSGLHLVKRR | SAMS-containing peptide as substrate | Brassica oleracea | ADP + ? | - |
? | |
ATP + HMGSAMSGLHLVKRR | SAMS-containing peptide as substrate | Brassica oleracea | ADP + ? | - |
? | |
ATP + HMHSAMSGLHLVKRR | - |
Brassica oleracea | ? | - |
? | |
ATP + HMKSAMSGLHLVKRR | synthetic SAMS-containing peptide as substrate | Brassica oleracea | ADP + ? | - |
? | |
ATP + HMRSAGSGLHLVKRR | SAMS-containing peptide as substrate | Brassica oleracea | ADP + ? | - |
? | |
ATP + HMRSAMSGLHGGKRR | SAMS-containing peptide as substrate | Brassica oleracea | ADP + ? | - |
? | |
ATP + HMRSAMSGLHGVKRR | SAMS-containing peptide as substrate | Brassica oleracea | ADP + ? | - |
? | |
ATP + HMRSAMSGLHLGKRR | SAMS-containing peptide as substrate | Brassica oleracea | ADP + ? | - |
? | |
ATP + HMRSAMSGLHLVKRR | SAMS-containing peptide as substrate | Brassica oleracea | ADP + ? | - |
? | |
ATP + HMRSAMTGLHGVKRR | - |
Brassica oleracea | ? | - |
? | |
ATP + HMRSAMTGLHLVKRR | SAMS-containing peptide as substrate | Brassica oleracea | ADP + ? | - |
? | |
ATP + HMRSAMYGLHLVKRR | SAMS-containing peptide as substrate | Brassica oleracea | ADP + ? | - |
? | |
ATP + [hydroxymethylglutaryl-CoA reductase (NADPH)] | 2 isoforms, major form A and minor form B, both phosphorylates mammalian HMG-CoA reductase | Brassica oleracea | ADP + [hydroxymethylglutaryl-CoA reductase (NADPH)] phosphate | - |
? | |
ATP + [hydroxymethylglutaryl-CoA reductase (NADPH)] | inactivates EC 1.1.1.34 by phosphorylation | Brassica oleracea | ADP + [hydroxymethylglutaryl-CoA reductase (NADPH)] phosphate | - |
? |
Subunits | Comment | Organism |
---|---|---|
? | x * 58000, catalytic subunit | Brassica oleracea |