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Literature summary for 2.7.11.26 extracted from

  • Manceur, A.P.; Driscoll, B.D.; Sun, W.; Audet, J.
    Selective enhancement of the uptake and bioactivity of a TAT-conjugated peptide inhibitor of glycogen synthase kinase-3 (2009), Mol. Ther., 17, 500-507.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
(2'Z,3'E)-6-bromoindirubin-3'-oxime
-
Homo sapiens
(2'Z,3'E)-6-bromoindirubin-3'-oxime
-
Mus musculus
lithium
-
Homo sapiens
lithium
-
Mus musculus
trans-activating transcriptor-eIF2B acts as a competitive inhibitor of GSK-3 Homo sapiens
trans-activating transcriptor-eIF2B acts as a competitive inhibitor of GSK-3 Mus musculus

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
bone marrow
-
Mus musculus
-
embryonic stem cell
-
Mus musculus
-
primary cell
-
Mus musculus
-
R1 ES cell
-
Mus musculus
-
TF-1 cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + beta-catenin
-
Mus musculus ADP + phosphorylated beta-catenin
-
?
ATP + beta-catenin
-
Homo sapiens ADP + phosphorylated beta-catenin
-
?
ATP + eIF2B peptide
-
Mus musculus ADP + phosphorylated eIF2B peptide
-
?
ATP + eIF2B peptide
-
Homo sapiens ADP + phosphorylated eIF2B peptide
-
?

Synonyms

Synonyms Comment Organism
glycogen synthase kinase-3
-
Mus musculus
glycogen synthase kinase-3
-
Homo sapiens
GSK-3
-
Mus musculus
GSK-3
-
Homo sapiens

Cofactor

Cofactor Comment Organism Structure
ATP
-
Mus musculus
ATP
-
Homo sapiens