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BRENDA support

Literature summary for 2.7.11.26 extracted from

  • Resende, R.; Ferreiro, E.; Pereira, C.; Oliveira, C.R.
    ER stress is involved in Abeta-induced GSK-3beta activation and tau phosphorylation (2008), J. Neurosci. Res., 86, 2091-2099.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
amyloid-beta 1-42 peptide 0.005 mM Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
dantrolene in the presence of dantrolene, GSK-3beta activation and tau phosphorylation are decreased Rattus norvegicus
GSK3betaI 0.0001 mM Rattus norvegicus
LiCl 10 mM Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
cerebral cortical neuron
-
Rattus norvegicus
-
primary culture
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + protein tau
-
Rattus norvegicus ADP + protein tau phosphate
-
?

Synonyms

Synonyms Comment Organism
glycogen synthase kinase-3beta
-
Rattus norvegicus
GSK-3beta
-
Rattus norvegicus

Cofactor

Cofactor Comment Organism Structure
ATP
-
Rattus norvegicus