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Literature summary for 2.7.11.18 extracted from

  • Leveille, N.; Fournier, A.; Labrie, C.
    Androgens down-regulate myosin light chain kinase in human prostate cancer cells (2009), J. Steroid Biochem. Mol. Biol., 114, 174-179.
    View publication on PubMed

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
breast cancer cell
-
Homo sapiens
-
CAMA-1 cell
-
Homo sapiens
-
DU-145 cell
-
Homo sapiens
-
LNCaP cell LNCaP cells express both long (non-muscle) and short (smooth muscle) isoforms of MLCK Homo sapiens
-
MDA-MB-231 cell
-
Homo sapiens
-
PC-3 cell
-
Homo sapiens
-
prostate cancer cell line
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + myosin light chain
-
Homo sapiens ADP + myosin light chain phosphate
-
?

Synonyms

Synonyms Comment Organism
MLCK
-
Homo sapiens
myosin light chain kinase
-
Homo sapiens

Cofactor

Cofactor Comment Organism Structure
ATP
-
Homo sapiens

Expression

Organism Comment Expression
Homo sapiens 0.1 nM androgen R1881 causes a progressive decrease in MLCK mRNA levels which decreases by 70% and 90%, respectively, at 24 and 48 h down