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Literature summary for 2.7.11.15 extracted from

  • Xin, W.; Tran, T.M.; Richter, W.; Clark, R.B.; Rich, T.C.
    Roles of GRK and PDE4 activities in the regulation of beta2 adrenergic signaling (2008), J. Gen. Physiol., 131, 349-364.
    View publication on PubMedView publication on EuropePMC

Inhibitors

Inhibitors Comment Organism Structure
59-74E
-
Homo sapiens

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
additional information
-
additional information kinetics Homo sapiens

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + beta2-adrenergic receptor Homo sapiens role of GRK activity in the regulation of beta2 adrenergic signaling, feedback mechanism, overview ADP + beta2-adrenergic receptor phosphate
-
?
additional information Homo sapiens GRK-mediated desensitization of beta2-adrenergic receptors is sufficient to cause declines in cAMP signals. GRK-mediated desensitization is primarily responsible for a sustained suppression of beta2AR signaling, overview ?
-
?

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
HEK-293 cell
-
Homo sapiens
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + beta2-adrenergic receptor
-
Homo sapiens ADP + beta2-adrenergic receptor phosphate
-
?
ATP + beta2-adrenergic receptor role of GRK activity in the regulation of beta2 adrenergic signaling, feedback mechanism, overview Homo sapiens ADP + beta2-adrenergic receptor phosphate
-
?
additional information GRK-mediated desensitization of beta2-adrenergic receptors is sufficient to cause declines in cAMP signals. GRK-mediated desensitization is primarily responsible for a sustained suppression of beta2AR signaling, overview Homo sapiens ?
-
?

Cofactor

Cofactor Comment Organism Structure
ATP
-
Homo sapiens